A novel one-pot reaction of heterocyclic ketene aminals: Synthesis of a small library of tetrahydropyridinone-fused 1,3-diazaheterocycles

被引：70
作者：
Yu, Chu-Yi [1 ]
Yang, Peng-Hui
Zhao, Mei-Xin
Huang, Zhi-Tang
机构：
[1] Chinese Acad Sci, Inst Chem, Biol Chem Lab, BNLMS, Beijing 100080, Peoples R China
[2] Grad Univ, Chinese Acad Sci, Beijing 100049, Peoples R China
来源：
SYNLETT | 2006年 / 12期
关键词：
one-pot reaction; heterocyclic ketene aminals; tetrahydropyridinones; 1,3-diazaheterocycles; synthesis;
D O I：
10.1055/s-2006-947343
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Inspired by the concept of multicomponent reactions, a novel one-pot reaction involving heterocyclic ketene aminals (HKAs), Meldrum's acid and aldehydes has been developed and employed for the construction of a small library of tetrahydropyridinone-fused 1,3-diazaheterocycles.
引用
收藏
页码：1835 / 1840
页数：6
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