The synthesis and biological activities of N-(3-pyridylmethyl) N′-(trans-2-thio-4-substituted phenyl-5,5-dimethyl-1,3,2-dioxaphosphinane-2-yl)thioureas

被引:4
作者
Shi, De-Qing [1 ]
Feras, Abudhaim [1 ]
Hamdan, Y. [1 ]
Liu, Yi [1 ]
Tan, Xiao-Song [1 ]
机构
[1] Cent China Normal Univ, Coll Chem, Key Lab Pesticide & Chem Biol, Minist Educ, Wuhan 430079, Hubei, Peoples R China
基金
中国国家自然科学基金;
关键词
biological activity; 1,3,2-dioxaphosphinane; substituted pyridine; synthesis; thiourea;
D O I
10.1080/10426500500542968
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
A series of novel title compounds were synthesized by the addition reaction of trans 2-isothiocyano-4-substitutedphenyl-5,5-dimethyl-1,3,2-dioxaphosphinane-2-sulfide to 3-aminomethylpyridine or 2-chloro-5-amino methylpyridine. Their structures were confirmed by H-1 NMR, P-31 NMR, IR, MS, and elemental analyses. Results of preliminary bioassay showed that all new compounds possess good fungicidal activity and insecticidal activity to some extent.
引用
收藏
页码:1831 / 1838
页数:8
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