Synthesis and antimicrobial activities of some new 2-substituted benzoxazole/benzothiazole derivatives

被引:0
|
作者
ElShaaer, HM
AbdelAziz, SA
Allimony, HA
Ali, UF
AbdelRahman, RM
机构
[1] AIN SHAMS UNIV,FAC EDUC,DEPT CHEM,DIV ORGAN CHEM,CAIRO,EGYPT
[2] AIN SHAMS UNIV,FAC EDUC,DEPT BIOL & GEOL SCI,CAIRO,EGYPT
来源
PHARMAZIE | 1997年 / 52卷 / 08期
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D O I
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中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
In the search for new antimicrobial compounds, several new sulfur bearing heterobicyclic moieties (4-11) have been synthesized by acylation and alkylation of acetamide, thioacetamide and semicarbazide derivatives. The structure of the products was deduced from elemental analyses as well as spectral data (IR, H-1 NMR and MS). Significant antimicrobial activities were obtained for all new compounds especially against Fusarium oxysporum.
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页码:585 / 589
页数:5
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