Regioselective Synthesis of Pyrazoles and Isoxazoles with Cyclopropanated Side-Chain

被引：8

作者：

Bendrath, Franziska ^{[1
]}

Falodun, Abiodun ^{[2
]}

Abilov, Zharylkasyn A. ^{[3
]}

Villinger, Alexander ^{[1
]}

Langer, Peter ^{[1
,4
]}

机构：

[1] Univ Rostock, Inst Chem, D-18059 Rostock, Germany

[2] Univ Benin, Fac Pharm, Dept Pharmaceut Chem, Benin, Nigeria

[3] Al Farabi Kazakh Natl Univ, Alma Ata 050040, Kazakhstan

[4] Univ Rostock, Leibniz Inst Katalyse eV, D-18059 Rostock, Germany

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2014年 / 51卷 / 03期

关键词：

DERIVATIVES; ZONIPORIDE;

D O I：

10.1002/jhet.1960

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Pyrazoles and isoxazoles with cyclopropanated side-chain were prepared by cyclization of cyclopropanated 1,3,5-tricarbonyl compounds with hydrazine and hydroxylamine, respectively. The regioselectivity is influenced by the reaction conditions.

引用

页码：835 / 840

页数：6

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