Cu(I)-promoted one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles from anti-3-aryl-2,3-dibromopropanoic acids and nitrobenzaldehydes

被引:4
|
作者
Liu, Xia [1 ]
Su, Changhui [2 ]
机构
[1] Jiangsu Open Univ, Coll Environm & Ecol, Nanjing 210036, Jiangsu, Peoples R China
[2] Nanjing Univ, Jinling Coll, Sch Chem & Life Sci, Nanjing, Jiangsu, Peoples R China
基金
中国国家自然科学基金;
关键词
1,2,3-triazoles; anti-3-aryl-2,3-dibromopropanoic acid; click chemistry; one-pot; STEREOSELECTIVE-SYNTHESIS; TERMINAL ALKYNES; AZIDES; CYCLOADDITION;
D O I
10.1080/00397911.2016.1262039
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of 1,4-disubstituted 1,2,3-triazoles were synthesized through a one-pot process from easily available anti-3-aryl-2,3-dibromopropanoic acids and nitrobenzaldehydes in hexamethylphosphoric triamide. Inexpensive copper(I) iodide was the catalyst.
引用
收藏
页码:279 / 284
页数:6
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