共 50 条
- [1] Discovery of the First BRD4 Second Bromodomain (BD2)-Selective InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (23) : 21577 - 21616Li, Junhua论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaHu, Qingqing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaZhu, Run论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaDong, Ruibo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Jilin Univ, Sch Pharmaceut Sci, Changchun 130021, Jilin, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaShen, Hui论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaHu, Jiankang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaZhang, Cheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaZhang, Xiaohan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Guangzhou Inst Biomed & Hlth, Anal & Testing Ctr, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaXu, Tingting论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaXiang, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Guoke Ningbo Life Sci & Hlth Ind Res Inst, Ningbo 315010, Zhejiang, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaZhang, Yan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaLin, Bin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaZhao, Linxiang论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaWu, Xishan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R ChinaXu, Yong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China Shenyang Pharmaceut Univ, Key Lab Struct Based Drug Design & Discovery, Minist Educ, Shenyang 110016, Peoples R China Chinese Acad Sci, Inst Drug Discovery, Guangzhou Inst Biomed & Hlth, China New Zealand Joint Lab Biomed & Hlth,Guangdon, Guangzhou 510530, Peoples R China
- [2] Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probesEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 209Chen, Jingjing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaLi, Yalei论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaZhang, Jie论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaZhang, Minmin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaWei, Aihuan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaLiu, Hongchun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaXie, Zhicheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaRen, Wenming论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaDuan, Wenwen论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaZhang, Zhuo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaShen, Aijun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Div Antitumor Pharmacol, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R ChinaHu, Youhong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 110039, Peoples R China UCAS, Sch Pharmaceut Sci & Technol, Hangzhou Inst Adv Study, Hangzhou 310024, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Dept Med Chem, State Key Lab Drug Res, 555 ZuChongZhi Rd, Shanghai 201203, Peoples R China
- [3] Discovery of novel small molecule induced selective degradation of the bromodomain and extra-terminal (BET) bromodomain protein BRD4 and BRD2 with cellular potenciesBIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (01)Jiang, Fei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaWei, Qingyun论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Affiliated Hosp Integrated Tradit Chinese & Weste, Nanjing 210028, Jiangsu, Peoples R China Jiangsu Prov Acad Tradit Chinese Med, Lab Cellular & Mol Biol, 100 Cross St,Hongshan Rd, Nanjing 210028, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaLi, Huili论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaLi, Hongmei论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaCui, Yong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaMa, Yu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaChen, Haifang论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaCao, Peng论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Affiliated Hosp Integrated Tradit Chinese & Weste, Nanjing 210028, Jiangsu, Peoples R China Jiangsu Prov Acad Tradit Chinese Med, Lab Cellular & Mol Biol, 100 Cross St,Hongshan Rd, Nanjing 210028, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaLu, Tao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaChen, Yadong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China
- [4] JAK2 inhibition for the treatment of hematologic and solid malignanciesEXPERT OPINION ON INVESTIGATIONAL DRUGS, 2012, 21 (05) : 637 - 655Harry, Brian L.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Med Scientist Training Program, Aurora, CO 80045 USA Univ Colorado, Sch Med, Dev Therapeut Program, Div Med Oncol, Aurora, CO 80045 USAEckhardt, S. Gail论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Dev Therapeut Program, Div Med Oncol, Aurora, CO 80045 USAJimeno, Antonio论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Dev Therapeut Program, Div Med Oncol, Aurora, CO 80045 USA Univ Colorado, Sch Med, Dev Therapeut Program, Div Med Oncol, Aurora, CO 80045 USA
- [5] Selective Small Molecule Induced Degradation of the BET Bromodomain Protein BRD4ACS CHEMICAL BIOLOGY, 2015, 10 (08) : 1770 - 1777Zengerle, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, Scotland Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, ScotlandChan, Kwok-Ho论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, Scotland Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, ScotlandCiulli, Alessio论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, Scotland Univ Dundee, Div Biol Chem & Drug Discovery, Coll Life Sci, James Black Ctr, Dundee DD1 SEH, Scotland
- [6] Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput dockingBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (11) : 2493 - 2496Zhao, Hongtao论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Biochem, CH-8057 Zurich, SwitzerlandGartenmann, Lisa论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Biochem, CH-8057 Zurich, SwitzerlandDong, Jing论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Biochem, CH-8057 Zurich, SwitzerlandSpiliotopoulos, Dimitrios论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Biochem, CH-8057 Zurich, SwitzerlandCaflisch, Amedeo论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Biochem, CH-8057 Zurich, Switzerland
- [7] Jak2 Inhibitors: Rationale and Role as Therapeutic Agents in Hematologic MalignanciesCURRENT ONCOLOGY REPORTS, 2009, 11 (02) : 117 - 124Sayyah, Jacqueline论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USASayeski, Peter P.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Physiol & Funct Genom, Gainesville, FL 32610 USA
- [8] Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (12) : 3399 - 3405Borysko, Petro论文数: 0 引用数: 0 h-index: 0机构: Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineMoroz, Yurii S.论文数: 0 引用数: 0 h-index: 0机构: Natl Taras Shevchenko Univ Kyiv, Volodymyrska St 60, UA-01601 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineVasylchenko, Oleksandr V.论文数: 0 引用数: 0 h-index: 0机构: Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineHurmach, Vasyl V.论文数: 0 引用数: 0 h-index: 0机构: Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Natl Taras Shevchenko Univ Kyiv, Volodymyrska St 60, UA-01601 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineStarodubtseva, Anastasia论文数: 0 引用数: 0 h-index: 0机构: Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineStefanishena, Natalia论文数: 0 引用数: 0 h-index: 0机构: Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineNesteruk, Kateryna论文数: 0 引用数: 0 h-index: 0机构: Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineZozulya, Sergey论文数: 0 引用数: 0 h-index: 0机构: Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineKondratov, Ivan S.论文数: 0 引用数: 0 h-index: 0机构: Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Natl Ukrainian Acad Sci, Inst Bioorgan Chem & Petrochem, Murmanska St 1, UA-02660 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, UkraineGrygorenko, Oleksandr O.论文数: 0 引用数: 0 h-index: 0机构: Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine Natl Taras Shevchenko Univ Kyiv, Volodymyrska St 60, UA-01601 Kiev, Ukraine Bienta Enamine Ltd, Chervonotkatska St 78, UA-02094 Kiev, Ukraine
- [9] Jak2 inhibitors: Rationale and role as therapeutic agents in hematologic malignanciesCurrent Oncology Reports, 2009, 11 : 117 - 124Jacqueline Sayyah论文数: 0 引用数: 0 h-index: 0机构: University of Florida College of Medicine,Department of Physiology and Functional GenomicsPeter P. Sayeski论文数: 0 引用数: 0 h-index: 0机构: University of Florida College of Medicine,Department of Physiology and Functional Genomics
- [10] Fragment-Based Drug Discovery of 2-Thiazolidinones as Inhibitors of the Histone Reader BRD4 BromodomainJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (10) : 3833 - 3851Zhao, Lele论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaCao, Danyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaChen, Tiantian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaWang, Yingqing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Div Antitumor Pharmacol, State Key Lab Drug Res, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaMiao, Zehong论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Div Antitumor Pharmacol, State Key Lab Drug Res, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaXu, Yechun论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaChen, Wuyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaWang, Xin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaLi, Yardian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaDu, Zhiyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaXiong, Bing论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaLi, Jian论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Appl Phys, Shanghai 201204, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaXu, Chunyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Appl Phys, Shanghai 201204, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaZhang, Naixia论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaHe, Jianhua论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Appl Phys, Shanghai 201204, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R ChinaShen, Jingkang论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Dept Med Chem, Shanghai 201203, Peoples R China