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Muskawar, Prashant Narayan
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Bhagat, Pundlik Rambhau
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY,
2014, 81
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Aher, Sainath Babaji
论文数: 0 引用数: 0
h-index: 0
机构:
VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India

Muskawar, Prashant Narayan
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h-index: 0
机构:
VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India

Thenmozhi, K.
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h-index: 0
机构:
VIT Univ, Sch Adv Sci, Environm & Analyt Chem Div, Vellore 632014, Tamil Nadu, India VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India

Bhagat, Pundlik Rambhau
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h-index: 0
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VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India VIT Univ, Sch Adv Sci, Div Organ Chem, Vellore 632014, Tamil Nadu, India
[2]
Discovery of N-(4-(3-amino-1H-indazol-4-yl)phenyl)-N'-(2-fluoro-5-methylphenyl)urea (ABT-869), a 3-aminoindazole-based orally active multitargeted receptor tyrosine kinase inhibitor
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Dai, Yujia
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Ji, Zhiqin
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Ahmed, Asma A.
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Bouska, Jennifer J.
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Bousquet, Peter F.
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Glaser, Keith B.
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Harris, Christopher M.
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Hickman, Dean
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Guo, Jun
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Marcotte, Patrick A.
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Marsh, Kennan C.
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2007, 50 (07)
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Dai, Yujia
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Hartandi, Kresna
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Ji, Zhiqin
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Ahmed, Asma A.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Albert, Daniel H.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Bauch, Joy L.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Bouska, Jennifer J.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Bousquet, Peter F.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Cunha, George A.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Glaser, Keith B.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Harris, Christopher M.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Hickman, Dean
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Guo, Jun
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Li, Junling
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Marcotte, Patrick A.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Marsh, Kennan C.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Moskey, Maria D.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Martin, Ruth L.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Olson, Amanda M.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Osterling, Donald J.
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h-index: 0
机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Pease, Lori J.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Soni, Niru B.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Stewart, Kent D.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Stoll, Vincent S.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Tapang, Paul
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Reuter, David R.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Davidsen, Steven K.
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机构: Abbott Labs, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA

Michaelides, Michael R.
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DeSantis, Carol E.
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Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Lin, Chun Chieh
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Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Mariotto, Angela B.
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NCI, Div Canc Control & Populat Sci, Data Modeling Branch, Bethesda, MD 20892 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Siegel, Rebecca L.
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Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Stein, Kevin D.
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Amer Canc Soc, Behav Res Ctr, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Kramer, Joan L.
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Amer Canc Soc, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Alteri, Rick
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Amer Canc Soc, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Robbins, Anthony S.
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Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA

Jemal, Ahmedin
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Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA Amer Canc Soc, Surveillance & Hlth Serv Res, Atlanta, GA 30303 USA
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El-Nassan, Hala Bakr
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EVAN, GI
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BROWN, L
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机构: Imperial Cancer Research Fund Laboratories, London, WC2A 3PX

WHYTE, M
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机构: Imperial Cancer Research Fund Laboratories, London, WC2A 3PX

HARRINGTON, E
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The identification of 2-(1H-indazol-4-yl)-6-(4-methanesulfonyl-piperazin-1-ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidine (GDC-0941) as a potent, selective, orally bioavailable inhibitor of class I PI3 kinase for the treatment of cancer
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Folkes, Adrian J.
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Alix, Sonia
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Baker, Stewart J.
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Box, Gary
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Chuckowree, Irina S.
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Clarke, Paul A.
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Depledge, Paul
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Eccles, Suzanne A.
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Friedman, Lori S.
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Hayes, Angela
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Hancox, Timothy C.
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Kugendradas, Arumugam
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Lensun, Letitia
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Moore, Pauline
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Olivero, Alan G.
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Pang, Jodie
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Patel, Sonal
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Robson, Anthony
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Folkes, Adrian J.
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Ahmadi, Khatereh
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h-index: 0
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Alderton, Wendy K.
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h-index: 0
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Alix, Sonia
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h-index: 0
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Baker, Stewart J.
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Box, Gary
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Chuckowree, Irina S.
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Clarke, Paul A.
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Depledge, Paul
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Eccles, Suzanne A.
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Friedman, Lori S.
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机构:
Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Hayes, Angela
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h-index: 0
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Hancox, Timothy C.
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Kugendradas, Arumugam
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Lensun, Letitia
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Moore, Pauline
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Olivero, Alan G.
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Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Pang, Jodie
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机构:
Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Patel, Sonal
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Pergl-Wilson, Giles H.
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Raynaud, Florence I.
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Robson, Anthony
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Saghir, Nahid
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h-index: 0
机构:
Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Salphati, Laurent
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Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Sohal, Sukhjit
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Piramed Pharma, Slough SL1 4NL, Berks, England Piramed Pharma, Slough SL1 4NL, Berks, England

Ultsch, Mark H.
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Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Valenti, Melanie
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Canc Res UK, Ctr Canc Therapeut, Inst Canc Res, Haddon Labs, Surrey SN2 5NG, England Piramed Pharma, Slough SL1 4NL, Berks, England

Wallweber, Heidi J. A.
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Genentech Inc, San Francisco, CA 94080 USA Piramed Pharma, Slough SL1 4NL, Berks, England

Wan, Nan Chi
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Wiesmann, Christian
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Workman, Paul
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Zhyvoloup, Alexander
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Zvelebil, Marketa J.
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Inst Canc Res, Breakthrough Breast Canc Res Ctr, London SW3 6JB, England Piramed Pharma, Slough SL1 4NL, Berks, England

Shuttleworth, Stephen J.
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Berry, Megan
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h-index: 0
机构:
Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Mathieu, Simon
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Nonomiya, Jim
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Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Olivero, Alan
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Pang, Jodie
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Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Peterson, David
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Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Salphati, Laurent
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Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Sampath, Deepak
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Genentech Inc, Small Mol Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Sideris, Steve
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Genentech Inc, Biochem Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Sutherlin, Daniel P.
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Tsui, Vickie
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Wan, Nan Chi
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Piramed Pharma, Slough SL1 4NL, Berks, England Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Wang, Shumei
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Wong, Susan
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Genentech Inc, Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA

Zhu, Bing-yan
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Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Discovery Chem, San Francisco, CA 94080 USA