Tropisetron inhibits the antinociceptive effect of intrathecally administered paracetamol and serotonin

被引:29
作者
Alloui, A [1 ]
Pelissier, T [1 ]
Dubray, C [1 ]
Lavarenne, J [1 ]
Eschalier, A [1 ]
机构
[1] FAC MED,DEPT FARMACOL,SANTIAGO 7,CHILE
关键词
paracetamol; nociception; serotonin; spinal cord; rats;
D O I
10.1111/j.1472-8206.1996.tb00593.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:406 / 407
页数:2
相关论文
共 8 条
[1]   ACETAMINOPHEN BLOCKS SPINAL HYPERALGESIA INDUCED BY NMDA AND SUBSTANCE-P [J].
BJORKMAN, R ;
HALLMAN, KM ;
HEDNER, J ;
HEDNER, T ;
HENNING, M .
PAIN, 1994, 57 (03) :259-264
[2]   THE 5-HT4 RECEPTOR - NAUGHTY, BUT NICE [J].
CLARKE, DE ;
CRAIG, DA ;
FOZARD, JR .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1989, 10 (10) :385-386
[3]   INHIBITION OF PROSTAGLANDIN SYNTHETASE IN BRAIN EXPLAINS ANTIPYRETIC ACTIVITY OF PARACETAMOL (4-ACETAMIDOPHENOL) [J].
FLOWER, RJ ;
VANE, JR .
NATURE, 1972, 240 (5381) :410-&
[4]   REVERSAL OF THE ANTINOCICEPTIVE EFFECTS OF INTRATHECALLY ADMINISTERED SEROTONIN IN THE RAT BY A SELECTIVE 5-HT3 RECEPTOR ANTAGONIST [J].
GLAUM, SR ;
PROUDFIT, HK ;
ANDERSON, EG .
NEUROSCIENCE LETTERS, 1988, 95 (1-3) :313-317
[5]   IDENTIFICATION OF 5-HT3 BINDING-SITES IN RAT SPINAL-CORD SYNAPTOSOMAL MEMBRANES [J].
GLAUM, SR ;
ANDERSON, EG .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 156 (02) :287-290
[6]  
MALMBERG AB, 1992, J PHARMACOL EXP THER, V263, P135
[7]   EVIDENCE OF A CENTRAL ANTINOCICEPTIVE EFFECT OF PARACETAMOL INVOLVING SPINAL 5HT(3) RECEPTORS [J].
PELISSIER, T ;
ALLOUI, A ;
PAEILE, C ;
ESCHALIER, A .
NEUROREPORT, 1995, 6 (11) :1546-1548
[8]   ANTINOCICEPTIVE EFFECT OF PARACETAMOL IN RATS IS PARTLY DEPENDENT ON SPINAL SEROTONERGIC SYSTEMS [J].
TJOLSEN, A ;
LUND, A ;
HOLE, K .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 193 (02) :193-201