Trans-diastereoselective synthesis of 3-phthalimido beta-lactams via a two step-Staudinger reaction.

被引：25
作者：
Bandini, E
Martelli, G
Spunta, G
Bongini, A
Panunzio, M
机构：
[1] CNR,ICOCEA,I-40129 BOLOGNA,ITALY
[2] UNIV BOLOGNA,I-40126 BOLOGNA,ITALY
[3] CNR,CTR STUDIO FIS MACROMOLEC,DIP CIAMICIAN,I-40126 BOLOGNA,ITALY
来源：
TETRAHEDRON LETTERS | 1996年 / 37卷 / 25期
关键词：
D O I：
10.1016/0040-4039(96)00841-6
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New conditions for the Staudinger reaction provide N-unsubstituted-3-phthalimido-beta-lactams in satisfactory yields with complete trans-selectivity. Copyright (C) 1996 Elsevier science Ltd
引用
收藏
页码：4409 / 4412
页数：4
相关论文
共 23 条
[1]   BETA-LACTAMS FROM ESTER ENOLATES AND SILYLIMINES - ENANTIOSELECTIVE SYNTHESIS OF THE TRANS-CARBAPENEM ANTIBIOTICS (+)-PS-5 AND (+)-PS-6 [J].
ANDREOLI, P ;
CAINELLI, G ;
PANUNZIO, M ;
BANDINI, E ;
MARTELLI, G ;
SPUNTA, G .
JOURNAL OF ORGANIC CHEMISTRY, 1991, 56 (21) :5984-5990
[2]   BETA-LACTAMS FROM ESTER ENOLATES AND SILYLIMINES - AN ENANTIOSPECIFIC SYNTHESIS OF MONOCYCLIC BETA-LACTAMS [J].
ANDREOLI, P ;
BILLI, L ;
CAINELLI, G ;
PANUNZIO, M ;
BANDINI, E ;
MARTELLI, G ;
SPUNTA, G .
TETRAHEDRON, 1991, 47 (43) :9061-9070
[3]   SYNTHESIS OF CARBAPENEMS VIA METALLOIMINES-ESTER ENOLATES CONDENSATION - A NEW SYNTHESIS OF (+)-1-BETA-METHYL PS-5 [J].
BANDINI, E ;
CAINELLI, G ;
GIACOMINI, D ;
MARTELLI, G ;
PANUNZIO, M ;
SPUNTA, G .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (11) :2347-2350
[4]  
BANDINI E, 1993, GAZZ CHIM ITAL, V123, P509
[5]  
BIRKOFER L, 1977, LIEBIGS ANN CHEM, P760
[6]  
BONANOMI G, 1996, TETRAHEDRON LETT, V37, P2467
[7]   CYCLO-ADDITIONS OF (ALKYLARYLAMINO)KETENES WITH IMINES - CIS-3-AMINO-2-AZETIDINONES [J].
BRADY, WT ;
GU, YQ .
JOURNAL OF ORGANIC CHEMISTRY, 1989, 54 (12) :2838-2842
[8]   Diastereofacial selectivity in the reaction of chiral N-trimethylsilyl imines with ester enolates: Preparation of trans-azetidin-2-ones in high stereocontrolled fashion [J].
Cainelli, G ;
Panunzio, M ;
Bandini, E ;
Martelli, G ;
Spunta, G .
TETRAHEDRON, 1996, 52 (05) :1685-1698
[9]   BETA-LACTAMS FROM ESTER ENOLATES AND N-TMSIMINES - ENANTIOSELECTIVE SYNTHESIS OF (6R,7S)-1-BETA-3-DIMETHYL-3-ISOCEPHEM [J].
CAINELLI, G ;
PANUNZIO, M ;
BANDINI, E ;
MARTELLI, G ;
SPUNTA, G ;
DACOL, M .
TETRAHEDRON, 1995, 51 (17) :5067-5072
[10]  
CAINELLI G, 1991, FARMACO, V46, P177
123