A convenient synthesis of 6-substituted-2,2-dimethyl-2H-1-benzopyrans

被引：10

作者：

Ding, CZ

机构：

[1] Bristol-Myers Squibb P., Princeton, NJ 08543-4000

来源：

SYNTHETIC COMMUNICATIONS | 1996年 / 26卷 / 22期

关键词：

D O I：

10.1080/00397919608004664

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Various 2,2-dimethyl-6-functional-2H-1-benzopyrans were prepared via a halogen-metal exchange reaction followed by treatment with electrophiles. These 6-functionalized chromenes are important synthetic intermediates for preparation of benzopyran-based potassium channel openers.

引用

页码：4267 / 4273

页数：7

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