Anxiolytic-like properties of ONO-9270578, a novel TRPC4/5 inhibitor, in mice

被引:0
作者
Kishi, A. [1 ]
Niwa, T. [1 ]
Kitajima, T. [1 ]
Kamimura, Y. [2 ]
Sasamura, T. [2 ]
Hirohka, T. [3 ]
Saitou, T. [3 ]
Katsumata, S. [1 ]
机构
[1] ONO Pharmaceut Co Itd, Discovery Res Labs, Osaka, Japan
[2] ONO Pharmaceut Co Itd, Exploratory Res Labs, Osaka, Japan
[3] ONO Pharmaceut Co Itd, Med Chem Res Labs, Osaka, Japan
关键词
CHANNELS; BEHAVIOR; AMYGDALA;
D O I
10.1016/S0924-977X(16)31667-4
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
P.4.a.005
引用
收藏
页码:S595 / S595
页数:1
相关论文
共 5 条
[1]   Emerging Roles of Canonical TRP Channels in Neuronal Function [J].
Bollimuntha, Sunitha ;
Selvaraj, Senthil ;
Singh, Brij B. .
TRANSIENT RECEPTOR POTENTIAL CHANNELS, 2011, 704 :573-593
[2]   MOLECULAR CHARACTERIZATION OF THE DROSOPHILA TRP LOCUS - A PUTATIVE INTEGRAL MEMBRANE-PROTEIN REQUIRED FOR PHOTOTRANSDUCTION [J].
MONTELL, C ;
RUBIN, GM .
NEURON, 1989, 2 (04) :1313-1323
[3]   The transient receptor potential family of ion channels [J].
Nilius, Bernd ;
Owsianik, Grzegorz .
GENOME BIOLOGY, 2011, 12 (03)
[4]   Decreased Anxiety-Like Behavior and Gαq/11-Dependent Responses in the Amygdala of Mice Lacking TRPC4 Channels [J].
Riccio, Antonio ;
Li, Yan ;
Tsvetkov, Evgeny ;
Gapon, Svetlana ;
Yao, Gui Lan ;
Smith, Kiersten S. ;
Engin, Elif ;
Rudolph, Uwe ;
Bolshakov, Vadim Y. ;
Clapham, David E. .
JOURNAL OF NEUROSCIENCE, 2014, 34 (10) :3653-3667
[5]   Essential Role for TRPC5 in Amygdala Function and Fear-Related Behavior [J].
Riccio, Antonio ;
Li, Yan ;
Moon, Jisook ;
Kim, Kwang-Soo ;
Smith, Kiersten S. ;
Rudolph, Uwe ;
Gapon, Svetlana ;
Yao, Gui Lan ;
Tsvetkov, Evgeny ;
Rodig, Scott J. ;
Van't Veer, Ashlee ;
Meloni, Edward G. ;
Carlezon, William A., Jr. ;
Bolshakov, Vadim Y. ;
Clapham, David E. .
CELL, 2009, 137 (04) :761-772