Asymmetric synthesis of stable α-aminoboronic esters catalyzed by N-heterocylic carbene and copper(I) chloride

[1] Asymmetric copper-catalyzed synthesis of α-amino boronate esters from N-tert-butanesulfinyl aldimines[J]. Beenen, Melissa A.;An, Chihui;Ellman, Jonathan A. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2008(22)

[2] Böhm VPW, 2001, ANGEW CHEM INT EDIT, V40, P3387

[3] Dipeptide boronic acid inhibitors of dipeptidyl peptidase IV: Determinants of potency and in vivo efficacy and safety[J]. Connolly, Beth A.;Sanford, David G.;Chiluwal, Amrita K.;Healey, Sarah E.;Peters, Diane E.;Dimare, Matthew T.;Wu, Wengen;Liu, Yuxin;Maw, Hlaing;Zhou, Yuhong;Li, Youhua;Jin, Zhiping;Sudmeier, James L.;Lai, Jack H.;Bachovchin, William W. JOURNAL OF MEDICINAL CHEMISTRY, 2008(19)

[4] Dalla Via L, 2012, FUTURE MED CHEM, V4, P525, DOI [10.4155/FMC.11.187, 10.4155/fmc.11.187]

[5] The first applications of carbene ligands in cross-couplings of alkyl electrophiles: Sonogashira reactions of unactivated alkyl bromides and iodides[J]. Eckhardt, M;Fu, GC. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2003(45)

[6] The 26S proteasome complex: An attractive target for cancer therapy[J]. Frankland-Searby, Sarah;Bhaumik, Sukesh R. BIOCHIMICA ET BIOPHYSICA ACTA-REVIEWS ON CANCER, 2012(01)

[7] Palladium/imidazolium salt catalyzed coupling of aryl halides with hypervalent organostannates[J]. Grasa, GA;Nolan, SP. ORGANIC LETTERS, 2001(01)

[8] Herrmann WA, 1998, J ORGANOMET CHEM, V557, P93

[9] N-Heterocyclic Carbene Catalysis: Enantioselective Formal [2+2] Cycloaddition of Ketenes and N-Sulfinylanilines[J]. Jian, Teng-Yue;He, Lin;Tang, Cen;Ye, Song. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2011(39)

[10] Proteasome Inhibitors: An Expanding Army Attacking a Unique Target[J]. Kisselev, Alexei F.;van der Linden, Wouter A.;Overkleeft, Herman S. CHEMISTRY & BIOLOGY, 2012(01)

[1] Asymmetric copper-catalyzed synthesis of α-amino boronate esters from N-tert-butanesulfinyl aldimines[J]. Beenen, Melissa A.;An, Chihui;Ellman, Jonathan A. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2008(22)

[2] Böhm VPW, 2001, ANGEW CHEM INT EDIT, V40, P3387

[3] Dipeptide boronic acid inhibitors of dipeptidyl peptidase IV: Determinants of potency and in vivo efficacy and safety[J]. Connolly, Beth A.;Sanford, David G.;Chiluwal, Amrita K.;Healey, Sarah E.;Peters, Diane E.;Dimare, Matthew T.;Wu, Wengen;Liu, Yuxin;Maw, Hlaing;Zhou, Yuhong;Li, Youhua;Jin, Zhiping;Sudmeier, James L.;Lai, Jack H.;Bachovchin, William W. JOURNAL OF MEDICINAL CHEMISTRY, 2008(19)

[4] Dalla Via L, 2012, FUTURE MED CHEM, V4, P525, DOI [10.4155/FMC.11.187, 10.4155/fmc.11.187]

[5] The first applications of carbene ligands in cross-couplings of alkyl electrophiles: Sonogashira reactions of unactivated alkyl bromides and iodides[J]. Eckhardt, M;Fu, GC. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2003(45)

[6] The 26S proteasome complex: An attractive target for cancer therapy[J]. Frankland-Searby, Sarah;Bhaumik, Sukesh R. BIOCHIMICA ET BIOPHYSICA ACTA-REVIEWS ON CANCER, 2012(01)

[7] Palladium/imidazolium salt catalyzed coupling of aryl halides with hypervalent organostannates[J]. Grasa, GA;Nolan, SP. ORGANIC LETTERS, 2001(01)

[8] Herrmann WA, 1998, J ORGANOMET CHEM, V557, P93

[9] N-Heterocyclic Carbene Catalysis: Enantioselective Formal [2+2] Cycloaddition of Ketenes and N-Sulfinylanilines[J]. Jian, Teng-Yue;He, Lin;Tang, Cen;Ye, Song. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2011(39)

[10] Proteasome Inhibitors: An Expanding Army Attacking a Unique Target[J]. Kisselev, Alexei F.;van der Linden, Wouter A.;Overkleeft, Herman S. CHEMISTRY & BIOLOGY, 2012(01)