Reaction of 3-aminocyclohex-2-en-1-ones with arylidenemalononitriles: Synthesis of N-substituted 1,4,5,6,7,8-hexahydroquinolin-5-ones

被引：15

作者：

Lichitsky, BV ^{[1
]}

Dudinov, AA ^{[1
]}

Krayushkin, MM ^{[1
]}

机构：

[1] Russian Acad Sci, ND Zelinskii Organ Chem Inst, 47 Leninsky Prosp,GSP-1, Moscow 119991, Russia

来源：

ARKIVOC | 2001年 / 2卷

关键词：

3-aminocyclohex-2-en-1-ones; 3-hydrazinocyclohex-2-en-1-ones; 2-arylidene-malononitriles; 1,4,5,6,7,8-hexahydroquinolin-5-ones;

D O I：

10.3998/ark.5550190.0002.911

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of 3-amino- and 3-hydrazinocyclohex-2-en-1-ones derived from cyclohexane-1,3-diones and an appropriate amine or hydrazine with 2-arylidenemalononitriles was investigated. An efficient method for the synthesis of N-substituted 1,4,5,6,7,8-hexahydroquinolin-5-ones was elaborated.

引用

页码：73 / 79

页数：7

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