A transgenic mouse model for in vivo regulation of the human CYP3A4 promoter

被引:0
作者
Zhang, WS [1 ]
Purchio, A [1 ]
Chen, K [1 ]
Wu, JM [1 ]
Lu, L [1 ]
West, DB [1 ]
机构
[1] Xenogen Corp, Alameda, CA 94501 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
235
引用
收藏
页码:118 / 118
页数:1
相关论文
共 50 条
  • [41] Contribution of metabolites to in vivo CYP3A4 inhibition by itraconazole
    Templeton, Ian E.
    Thummel, Kenneth E.
    Isoherranen, Nina
    Kharasch, Evan David
    Kunze, Kent L.
    Nelson, Wendel L.
    Hoffer, Christine
    DRUG METABOLISM REVIEWS, 2006, 38 : 127 - 128
  • [42] CYP3A4 HUMANIZED MOUSE; A MODEL TO STUDY CYP3A4-MEDIATED DRUG-DRUG INTERACTION POTENTIAL
    Rose, Anne
    Xu, Carrie
    Johnghar, Susan
    Behnia, Kamelia
    DRUG METABOLISM REVIEWS, 2012, 44 : 76 - 77
  • [43] Molecular mechanism of the regulation of CYP3A4 by HNF4α
    Tegude, H
    Eichelbaum, M
    Burk, O
    DRUG METABOLISM REVIEWS, 2003, 35 : 144 - 144
  • [44] Detection of MboII polymorphism at the 5′ promoter region of CYP3A4
    Cavalli, SA
    Hirata, MH
    Hirata, RDC
    CLINICAL CHEMISTRY, 2001, 47 (02) : 348 - 351
  • [45] A Useful Model Capable of Predicting the Clearance of Cytochrome P450 3A4 (CYP3A4) Substrates in Humans: Validity of CYP3A4 Transgenic Mice Lacking Their Own Cyp3a Enzymes
    Mitsui, Tetsuya
    Nemoto, Takayuki
    Miyake, Taiji
    Nagao, Shunsuke
    Ogawa, Kotaro
    Kato, Motohiro
    Ishigai, Masaki
    Yamada, Hideyuki
    DRUG METABOLISM AND DISPOSITION, 2014, 42 (09) : 1540 - 1547
  • [46] Regulation of CYP3A4 expression by PAR transcription factors
    Mantei, Kristen E.
    Le, Min
    Klick, David E.
    Vyhlidal, Carrie A.
    Hines, Ronald N.
    FASEB JOURNAL, 2007, 21 (06) : A1183 - A1183
  • [47] Expression of CYP3A4 in human breast tumors
    Coban, T
    Kapucuoglu, N
    Raunio, H
    Pelkonen, O
    Edwards, RJ
    Boobis, AR
    Iscan, M
    DRUG METABOLISM REVIEWS, 2004, 36 : 92 - 92
  • [48] Receptor-dependent regulation of the CYP3A4 gene
    Gibson, G
    El-Sankary, W
    Bombail, V
    Plan, N
    TOXICOLOGY, 2001, 164 (1-3) : 15 - 15
  • [49] HUMAN PCIS AS EX VIVO MODEL TO STUDY THE INTERPLAY BETWEEN P-GP AND CYP3A4 IN THE INTESTINE
    Li, Ming
    de Graaf, Inge A. M.
    de Jager, Marina H.
    Groothuis, Geny M. M.
    DRUG METABOLISM REVIEWS, 2015, 47 : 164 - 165
  • [50] Transcriptional regulation of CYP3A4 by microtubule stabilizing drugs
    Mani, S
    Sundarababu, S
    Liu, WJ
    Ganjam, K
    Horwitz, SB
    DRUG METABOLISM REVIEWS, 2004, 36 : 302 - 302