Identification by site-directed mutagenesis of residues involved in ligand recognition and activation of human A3 adenosine receptors

被引:0
|
作者
Gaul, ZG
Chen, A
Barak, D
Kim, SK
Müller, CF
Jacobson, KA
机构
[1] NIDDK, Mol Recognit Sect, LBC, NIH, Bethesda, MD 20892 USA
[2] Univ Bonn, Inst Pharmaceut, D-5300 Bonn, Germany
关键词
D O I
暂无
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
107
引用
收藏
页码:566 / 566
页数:1
相关论文
共 50 条
  • [21] SITE-DIRECTED MUTAGENESIS OF ALPHA-2A-ADRENERGIC RECEPTORS - IDENTIFICATION OF AMINO-ACIDS INVOLVED IN LIGAND-BINDING AND RECEPTOR ACTIVATION BY AGONISTS
    WANG, CD
    BUCK, MA
    FRASER, CM
    MOLECULAR PHARMACOLOGY, 1991, 40 (02) : 168 - 179
  • [22] TRICHODIENE SYNTHASE - IDENTIFICATION OF ACTIVE-SITE RESIDUES BY SITE-DIRECTED MUTAGENESIS
    CANE, DE
    SHIM, JH
    XUE, Q
    FITZSIMONS, BC
    HOHN, TM
    BIOCHEMISTRY, 1995, 34 (08) : 2480 - 2488
  • [23] Site-directed mutagenesis of oxalate oxidase active-site residues involved in catalysis
    Grant, Morgan
    Hoffer, Eric
    Moomaw, Ellen
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242
  • [24] IDENTIFICATION OF RESIDUES ESSENTIAL FOR PROGESTERONE BINDING TO UTEROGLOBIN BY SITE-DIRECTED MUTAGENESIS
    PETER, W
    BRULLER, HJ
    VRIEND, G
    BEATO, M
    SUSKE, G
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1991, 38 (01): : 27 - 33
  • [25] Identification of lysine residues involved in electrostatic binding of the 33 kDa protein with PSII by site-directed mutagenesis
    Yuhi, K
    Suzuki, T
    Ohta, H
    Enami, I
    PLANT AND CELL PHYSIOLOGY, 2004, 45 : S80 - S80
  • [26] Identification of Critical Residues of the Mycobacterial Dephosphocoenzyme A Kinase by Site-Directed Mutagenesis
    Walia, Guneet
    Gajendar, Komatireddy
    Surolia, Avadhesha
    PLOS ONE, 2011, 6 (01):
  • [27] Site-directed mutagenesis of putative active site residues in human pyruvate dehydrogenase
    Korotchkina, LG
    Tripatara, A
    Ali, MS
    Patel, MS
    FASEB JOURNAL, 1997, 11 (09): : A890 - A890
  • [28] Site-directed mutagenesis of the human A(1) adenosine receptor: Influences of acidic and hydroxy residues in the first four transmembrane domains on ligand binding
    Barbhaiya, H
    McClain, R
    Ijzerman, A
    Rivkees, SA
    MOLECULAR PHARMACOLOGY, 1996, 50 (06) : 1635 - 1642
  • [29] Identification of residues involved in homotrimeric assembly of the human P2X4 receptor by simulations and site-directed mutagenesis
    Malisetty, Aparna Sai
    Schaffrath, Lukas
    Markwardt, Fritz
    Coenen, Saskia
    Machtens, Jan-Philipp
    Koeppen, Susan
    Schmalzing, Guenther
    BIOPHYSICAL JOURNAL, 2023, 122 (03) : 459A - 460A
  • [30] SITE-DIRECTED MUTAGENESIS AND BACTERIAL EXPRESSION OF HUMAN ADENOSINE-DEAMINASE
    DANTON, MJ
    LEONARDO, J
    RILEY, L
    COLEMAN, MS
    FEDERATION PROCEEDINGS, 1987, 46 (06) : 1985 - 1985