Rapid synthesis of oxazoles under microwave conditions

被引：65

作者：

Brain, CT ^{[1
]}

Paul, JM ^{[1
]}

机构：

[1] Novartis Inst Med Sci, London WC1E 6BN, England

来源：

SYNLETT | 1999年 / 10期

关键词：

oxazoles; cyclization; microwaves;

D O I：

10.1055/s-1999-2905

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new and efficient variation of the Robinson-Gabriel oxazole synthesis is described. Oxazoles were prepared by cyclodehydration of 2-acylamino carbonyl compounds with Burgess reagent under monomode microwave irradiation.

引用

页码：1642 / 1644

页数：3

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