Microwave-assisted synthesis of novel fluorinated 1,2,4-triazole derivatives, and study of their biological activity

被引:70
作者
Liu, Xing-Hai [1 ]
Weng, Jian-Quan [1 ]
Wang, Bao-Lei [2 ]
Li, Yong-Hong [2 ]
Tan, Cheng-Xia [1 ]
Li, Zheng-Ming [2 ]
机构
[1] Zhejiang Univ Technol, Coll Chem Engn & Mat Sci, Hangzhou 310014, Zhejiang, Peoples R China
[2] Nankai Univ, Natl Pesticidal Engn Ctr, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China
基金
中国国家自然科学基金;
关键词
1,2,4-Triazole; Fluorine; Herbicidal activity; Microwave irradiation synthesis; FUNGICIDAL ACTIVITY; CRYSTAL-STRUCTURE; CYCLOPROPANE MOIETY; 1,2,3-THIADIAZOLE; BIOACTIVITY;
D O I
10.1007/s11164-013-1113-4
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Microwave irradiation was used for synthesis of a series of novel fluorinated 1,2,4-triazole derivatives. The molecular structures of the compounds were determined by use of H-1 NMR and FTIR spectroscopy and MS and HRMS. Study of their biological activity showed most of the compounds had good herbicidal activity.
引用
收藏
页码:2605 / 2612
页数:8
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