A facile synthesis of benzo[b][1,4]thiazepine derivatives by palladium acetate catalyzed reaction

被引：13

作者：

Kaishap, Partha Pratim ^{[1
]}

Shekarrao, Kommuri ^{[1
]}

Saikia, Pallabi ^{[1
]}

Gogoi, Sanjib ^{[1
]}

Boruah, Romesh C. ^{[1
]}

机构：

[1] North East Inst Sci & Technol, Div Med Chem, Jorhat 785006, Assam, India

来源：

TETRAHEDRON LETTERS | 2014年 / 55卷 / 11期

关键词：

Benzo[b][1,4]thiazepine; Steroid; Palladium acetate; beta-Bromovinyl aldehyde; 2-Aminothiophenol; 1,3-DIPOLAR CYCLOADDITION; 1,5-BENZOTHIAZEPINES; QUINOLINES; PYRIDINE; SOLVENT;

D O I：

10.1016/j.tetlet.2014.01.153

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The preparation of steroid/nonsteroid fused benzo[b][1,4]thiazepines and 2-arylsubstituted benzo[b][1,4] thiazepines is described from Pd(OAc)(2) catalyzed reaction of steroidal/nonsteroidal beta-halovinyl aldehydes and 2-aminothiophenols in DMF under heating condition. (c) 2014 Elsevier Ltd. All rights reserved.

引用

页码：1927 / 1930

页数：4

共 22 条

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