Synthesis of 4,5,6-trisubstituted 3-cyanopyridine-2(1H)-thiones based on alpha-substituted beta-diketones

被引：2
|
作者：
Frolova, NG [1 ]
Zavyalova, VK [1 ]
Litvinov, VP [1 ]
机构：
[1] ND ZELINSKII INST ORGAN CHEM,MOSCOW 117913,RUSSIA
来源：
RUSSIAN CHEMICAL BULLETIN | 1996年 / 45卷 / 11期
关键词：
5-substituted 3-cyano-4,6-dimethylpyridine-2(1H)-thiones; cyanothioacetamide; cyclization; thieno[2,3-b]pyridines;
D O I：
10.1007/BF01431119
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
5-Substituted 3-cyano-4,6-dimethylpyridine-2(1H)-thiones were synthesized by the reaction of alpha-substituted beta-diketones with cyanothioacetamide in the presence of triethylamine. The compounds synthesized were converted into thieno[2,3-b]pyridines by treatment with organic halides and KOH.
引用
收藏
页码：2578 / 2580
页数：3
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