SYNTHESIS AND BIOLOGICAL ACTIVITY OF DELTORPHIN I AND DERMORPHIN ANALOGUES MODIFIED IN MESSAGE DOMAIN WITH NEW α,α-DISUBSTITUTED AMINO ACIDS

被引：0

作者：

Lasota, A. ^{[1
]}

Fraczak, O. ^{[1
]}

Olma, A. ^{[1
]}

Muchowska, A. ^{[2
]}

Lipkowski, A. ^{[2
]}

机构：

[1] Lodz Univ Technol, Inst Organ Chem, Lodz, Poland

[2] Polish Acad Sci, Mossakowski Med Res Ctr, Warsaw, Poland

来源：

JOURNAL OF PEPTIDE SCIENCE | 2014年 / 20卷

关键词：

opioid peptides; deltorphin; dermorphin; alpha; alpha-disubstitiuted amino acids; opioid receptor binding;

D O I：

暂无

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

P096

引用

页码：S171 / S171

页数：1

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[2] Dermorphin tetrapeptide analogs as potent and long-lasting analgesics with pharmacological profiles distinct from morphine [J].

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Sakurada, Tsukasa ;

Sakurada, Shinobu .

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[3] A convenient route to optically pure α-alkyl-β-(-amino)alanines [J].

Olma, A. ;

Lasota, A. ;

Kudaj, A. .

AMINO ACIDS, 2012, 42 (06) :2525-2528

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