AN EFFICIENT ONE-POT SYNTHESIS OF SOME NEW SUBSTITUTED 1,2,3,5-THIATRIAZOLIDIN-4-ONE 1,1-DIOXIDES

被引：2

作者：

Balti, Monaem ^{[1
]}

Dridi, Khaireddine ^{[1
]}

El Efrit, Mohamed Lotfi ^{[1
]}

机构：

[1] El Manar Univ, Coll Sci Tunis, Organ Chem Lab, Tunis, Tunisia

来源：

HETEROCYCLES | 2014年 / 89卷 / 06期

关键词：

1,2,5-THIADIAZOLIDIN-3-ONE 1,1 DIOXIDE; HIV-1 PROTEASE INHIBITORS; HUMAN-LEUKOCYTE ELASTASE; THIONYL CHLORIDE; SCAFFOLD; HETEROCYCLES; PROTEINASE-3; DERIVATIVES; DESIGN; AGENTS;

D O I：

10.3987/COM-14-12980

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of some new 1,2,3,5-thiatriazolidin-4-one 1,1-dioxides derivatives were synthesized by reacting respectively beta-cyanohydrazines and phosphorylated hydrazine with chlorosulfonyl isocyanate in good yields. The structures of all the newly prepared compounds were confirmed by IR, H-1, C-13, P-31-NMR spectral data and elemental analysis.

引用

页码：1483 / 1490

页数：8

共 26 条

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