Exploiting translation inhibition: antitumor efficacy of SVC112 in preclinical models of colorectal cancer

被引:0
|
作者
Robertson, Kelli M. [1 ]
Gustafson, Annika L. [1 ]
Tentler, John J. [1 ]
Bagby, Stacey M. [1 ]
Anna, Capasso [1 ]
Klauck, Peter J. [1 ]
Pitts, Todd M. [1 ]
Kim, Jihye [1 ]
Tan, Aik Choon [1 ]
Su, Tin Tin [2 ]
Eckhardt, S. Gail [1 ]
机构
[1] Univ Colorado, Sch Med, Denver, CO USA
[2] Univ Colorado, Denver, CO 80202 USA
关键词
D O I
10.1158/1535-7163.TARG-17-B051
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
B051
引用
收藏
页数:2
相关论文
共 50 条
  • [1] PRECLINICAL EVALUATION OF THE TRANSLATIONAL INHIBITOR SVC112 IN COLORECTAL CANCER
    Robertson, K.
    Tentler, J.
    Klauck, P.
    Bagby, S.
    Pitts, T.
    Kim, J.
    Eckhardt, S.
    JOURNAL OF INVESTIGATIVE MEDICINE, 2016, 64 (01) : 277 - 277
  • [2] Inhibiting Translation Elongation with SVC112 Suppresses Cancer Stem Cells and Inhibits Growth in Head and Neck Squamous Carcinoma
    Keysar, Stephen B.
    Gomes, Nathan
    Miller, Bettina
    Jackson, Brian C.
    Le, Phuong N.
    Morton, J. Jason
    Reisinger, Julie
    Chimed, Tugs-Saikhan
    Gomez, Karina E.
    Nieto, Cera
    Frederick, Barbara
    Pronk, Gijsbertus J.
    Somerset, Hilary L.
    Tan, Aik-Choon
    Wang, Xiao-Jing
    Raben, David
    Su, Tin Tin
    Jimeno, Antonio
    CANCER RESEARCH, 2020, 80 (05) : 1183 - 1198
  • [3] Synergistic antitumor activity of regorafenib and lapatinib in preclinical models of human colorectal cancer
    Zhang, Wen-Ji
    Li, Yong
    Wei, Meng-Ning
    Chen, Yao
    Qiu, Jian-Ge
    Jiang, Qi-Wei
    Yang, Yang
    Zheng, Di-Wei
    Qin, Wu-Ming
    Huang, Jia-Rong
    Wang, Kun
    Zhang, Wen-Juan
    Wang, Yi-Jun
    Yang, Dong-Hua
    Chen, Zhe-Sheng
    Shi, Zhi
    CANCER LETTERS, 2017, 386 : 100 - 109
  • [4] Defining efficacy thresholds in preclinical models of cancer: a comparative analysis of cetuximab efficacy and biomarkers in colorectal cancer models
    Prewett, M.
    Bassi, R.
    Paz, K.
    Amatulli, M.
    Samakoglu, S.
    Tonra, J. R.
    EJC SUPPLEMENTS, 2010, 8 (07): : 62 - 62
  • [5] Preclinical efficacy of carfilzomib in BRAF-mutant colorectal cancer models
    Maione, Federica
    Oddo, Daniele
    Galvagno, Federica
    Falcomata, Chiara
    Pandini, Marta
    Macagno, Marco
    Pessei, Valeria
    Barault, Ludovic
    Gigliotti, Chiara
    Mira, Alessia
    Corti, Giorgio
    Lamba, Simona
    Riganti, Chiara
    Castella, Barbara
    Massaia, Massimo
    Rad, Roland
    Saur, Dieter
    Bardelli, Alberto
    Di Nicolantonio, Federica
    MOLECULAR ONCOLOGY, 2024, 18 (06) : 1552 - 1570
  • [6] Efficacy of NEDD8 Pathway Inhibition in Preclinical Models of Poorly Differentiated, Clinically Aggressive Colorectal Cancer
    Picco, Gabriele
    Petti, Consalvo
    Sassi, Francesco
    Grillone, Katia
    Migliardi, Giorgia
    Rossi, Teresa
    Isella, Claudio
    Di Nicolantonio, Federica
    Sarotto, Ivana
    Sapino, Anna
    Bardelli, Alberto
    Trusolino, Livio
    Bertotti, Andrea
    Medico, Enzo
    JNCI-JOURNAL OF THE NATIONAL CANCER INSTITUTE, 2017, 109 (02):
  • [7] Mouse models of colorectal cancer as preclinical models
    McIntyre, Rebecca E.
    Buczacki, Simon J. A.
    Arends, Mark J.
    Adams, David J.
    BIOESSAYS, 2015, 37 (08) : 909 - 920
  • [8] Assessment of preclinical models for colorectal cancer
    Wilkinson, RW
    Ellison, D
    Poulsom, R
    Staub, J
    Ilyas, M
    Bodmer, WF
    Snary, D
    Mather, SJ
    Ross, EL
    BRITISH JOURNAL OF CANCER, 2001, 85 : 39 - 39
  • [9] Significant Therapeutic Efficacy with Combined Radioimmunotherapy and Cetuximab in Preclinical Models of Colorectal Cancer
    Vassileva, Vessela
    Rajkumar, Vineeth
    Mazzantini, Mario
    Robson, Mathew
    Badar, Adam
    Sharma, Surinder
    Arstad, Erik
    Hochhauser, Daniel
    Lythgoe, Mark F.
    Boxer, Geoffrey M.
    Pedley, Rosmund Barbara
    JOURNAL OF NUCLEAR MEDICINE, 2015, 56 (08) : 1239 - 1245
  • [10] Antitumor Activity of BRAF Inhibitor Vemurafenib in Preclinical Models of BRAF-Mutant Colorectal Cancer
    Yang, Hong
    Higgins, Brian
    Kolinsky, Kenneth
    Packman, Kathryn
    Bradley, William D.
    Lee, Richard J.
    Schostack, Kathleen
    Simcox, Mary Ellen
    Kopetz, Scott
    Heimbrook, David
    Lestini, Brian
    Bollag, Gideon
    Su, Fei
    CANCER RESEARCH, 2012, 72 (03) : 779 - 789