CrossTalk proposal: Weighing the evidence for Class A GPCR dimers, the evidence favours dimers

被引:48
作者
Bouvier, Michel [1 ]
Hebert, Terence E. [2 ]
机构
[1] Univ Montreal, IRIC, Dept Biochim, Montreal, PQ H3T 1J4, Canada
[2] McGill Univ, Dept Pharmacol & Therapeut, Montreal, PQ H3G 1Y6, Canada
来源
JOURNAL OF PHYSIOLOGY-LONDON | 2014年 / 592卷 / 12期
关键词
PROTEIN-COUPLED RECEPTORS; BINDING-PROPERTIES; MUSCARINIC RECEPTOR; OPIOID RECEPTOR; COMPLEX; RHODOPSIN; COOPERATIVITY; REVEALS; OLIGOMERIZATION; ORGANIZATION;
D O I
10.1113/jphysiol.2014.272252
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:2439 / 2441
页数:3
相关论文
共 30 条
[1]  
Albizu L, 2010, NAT CHEM BIOL, V6, P587, DOI [10.1038/NCHEMBIO.396, 10.1038/nchembio.396]
[2]   Heteromeric MT1/MT2 Melatonin Receptors Modulate Photoreceptor Function [J].
Baba, Kenkichi ;
Benleulmi-Chaachoua, Abla ;
Journe, Anne-Sophie ;
Kamal, Maud ;
Guillaume, Jean-Luc ;
Dussaud, Sebastien ;
Gbahou, Florence ;
Yettou, Katia ;
Liu, Cuimei ;
Contreras-Alcantara, Susana ;
Jockers, Ralf ;
Tosini, Gianluca .
SCIENCE SIGNALING, 2013, 6 (296)
[3]   Single-molecule analysis of fluorescently labeled G-protein-coupled receptors reveals complexes with distinct dynamics and organization [J].
Calebiro, Davide ;
Rieken, Finn ;
Wagner, Julia ;
Sungkaworn, Titiwat ;
Zabel, Ulrike ;
Borzi, Alfio ;
Cocucci, Emanuele ;
Zuern, Alexander ;
Lohse, Martin J. .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2013, 110 (02) :743-748
[4]   The apparent cooperativity of some GPCRs does not necessarily imply dimerization [J].
Chabre, Marc ;
Deterre, Philippe ;
Antonny, Bruno .
TRENDS IN PHARMACOLOGICAL SCIENCES, 2009, 30 (04) :182-187
[5]   Cardiac muscarinic receptors. Cooperativity as the basis for multiple states of affinity [J].
Chidiac, P ;
Green, MA ;
Pawagi, AB ;
Wells, JW .
BIOCHEMISTRY, 1997, 36 (24) :7361-7379
[6]   Fluorescent ligands to investigate GPCR binding properties and oligomerization [J].
Cottet, Martin ;
Faklaris, Orestis ;
Falco, Amadine ;
Trinquet, Eric ;
Pin, Jean-Philippe ;
Mouillac, Bernard ;
Durroux, Thierry .
BIOCHEMICAL SOCIETY TRANSACTIONS, 2013, 41 :148-153
[7]  
DELEAN A, 1980, J BIOL CHEM, V255, P7108
[8]   Instability of a Class A G Protein-Coupled Receptor Oligomer Interface [J].
Fonseca, Jacqueline M. ;
Lambert, Nevin A. .
MOLECULAR PHARMACOLOGY, 2009, 75 (06) :1296-1299
[9]   Atomic-force microscopy: Rhodopsin dimers in native disc membranes [J].
Fotiadis, D ;
Liang, Y ;
Filipek, S ;
Saperstein, DA ;
Engel, A ;
Palczewski, K .
NATURE, 2003, 421 (6919) :127-128
[10]   Decoding the Signaling of a GPCR Heteromeric Complex Reveals a Unifying Mechanism of Action of Antipsychotic Drugs [J].
Fribourg, Miguel ;
Moreno, Jose L. ;
Holloway, Terrell ;
Provasi, Davide ;
Baki, Lia ;
Mahajan, Rahul ;
Park, Gyu ;
Adney, Scott K. ;
Hatcher, Candice ;
Eltit, Jose M. ;
Ruta, Jeffrey D. ;
Albizu, Laura ;
Li, Zheng ;
Umali, Adrienne ;
Shim, Jihyun ;
Fabiato, Alexandre ;
MacKerell, Alexander D., Jr. ;
Brezina, Vladimir ;
Sealfon, Stuart C. ;
Filizola, Marta ;
Gonzalez-Maeso, Javier ;
Logothetis, Diomedes E. .
CELL, 2011, 147 (05) :1011-1023