Free radical method for the synthesis of spiro-piperidinyl heterocycles

被引：19
作者：
Chen, MH
Abraham, JA
机构：
[1] Department of Medicinal Chemistry, Merck Research Laboratories, Rahway, NJ 07065
[2] Harvard University, Cambridge, MA
来源：
TETRAHEDRON LETTERS | 1996年 / 37卷 / 30期
关键词：
D O I：
10.1016/0040-4039(96)01072-6
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A general approach to spiro-piperidinyl heterocycles (I, X=S, O, NH, NAc) was obtained from the key intermediate 3 via an efficient radical reaction. Copyright (C) 1996 Elsevier Science Ltd
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页码：5233 / 5234
页数：2
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