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- [1] Selective and Potent Morpholinone Inhibitors of the MDM2-p53 Protein-Protein InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (06) : 2472 - 2488Gonzalez, Ana Z.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAEksterowicz, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USABeck, Hilary P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAChow, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USADuquette, Jason论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAFox, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAFu, Jiasheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAHouze, Jonathan B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAJin, Lixia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALi, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALi, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALing, Yun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALong, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcGee, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcIntosh, Joel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcMinn, Dustin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USARew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAShaffer, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAWortman, Sarah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYakowec, Peter论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOlson, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA
- [2] Inhibitors of the MDM2-p53 interaction as anticancer drugsDRUGS OF THE FUTURE, 2007, 32 (10) : 883 - 896Hardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Northern Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Northern Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England
- [3] The MDM2-p53 interactionMOLECULAR CANCER RESEARCH, 2003, 1 (14) : 1001 - 1008Moll, UM论文数: 0 引用数: 0 h-index: 0机构: SUNY Stony Brook, Dept Pathol, Stony Brook, NY 11794 USA SUNY Stony Brook, Dept Pathol, Stony Brook, NY 11794 USAPetrenko, O论文数: 0 引用数: 0 h-index: 0机构: SUNY Stony Brook, Dept Pathol, Stony Brook, NY 11794 USA SUNY Stony Brook, Dept Pathol, Stony Brook, NY 11794 USA
- [4] Potent and Orally Active Small-Molecule Inhibitors of the MDM2-p53 InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (24) : 7970 - 7973Yu, Shanghai论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAQin, Dongguang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAShangary, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAChen, Jianyong论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Guoping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USADing, Ke论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAMcEachern, Donna论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAQiu, Su论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USANikolovska-Coleska, Zaneta论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAMiller, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAKang, Sanmao论文数: 0 引用数: 0 h-index: 0机构: Ascenta Therapeut Inc, Malvern, PA 19355 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAYang, Dajun论文数: 0 引用数: 0 h-index: 0机构: Ascenta Therapeut Inc, Malvern, PA 19355 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Dept Internal Med, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pharmacol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
- [5] Discovery of Potent and Simplified Piperidinone-Based Inhibitors of the MDM2-p53 InteractionACS MEDICINAL CHEMISTRY LETTERS, 2014, 5 (08): : 894 - 899Yu, Ming论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAWang, Yingcai论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAZhu, Jiang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAChow, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAEksterowicz, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAFox, Brian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAFu, Jiasheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAGribble, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALi, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALiu, Jiwen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALo, Mei-chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAMcMinn, Dustin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USARew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAShaffer, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOlson, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA
- [6] The development of piperidinones as potent MDM2-P53 protein - protein interaction inhibitors for cancer therapyEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 159 : 1 - 9Liao, Guochao论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaYang, Deying论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaMa, Leilei论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaLi, Wenwei论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaHu, Liqin论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaZeng, Liming论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaWu, Peng论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaDuan, Lixin论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaLiu, Zhongqiu论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China
- [7] Identification of substituted isoindolinones as potent inhibitors of the MDM2-p53 protein-protein interactionMOLECULAR CANCER THERAPEUTICS, 2009, 8 (12)Watson, Anna论文数: 0 引用数: 0 h-index: 0Liu, Junfeng论文数: 0 引用数: 0 h-index: 0Armstrong, Elizabeth论文数: 0 引用数: 0 h-index: 0Blackburn, Timothy论文数: 0 引用数: 0 h-index: 0Endicott, Jane A.论文数: 0 引用数: 0 h-index: 0Golding, Bernard T.论文数: 0 引用数: 0 h-index: 0Griffin, Roger J.论文数: 0 引用数: 0 h-index: 0Lu, Xiaohong论文数: 0 引用数: 0 h-index: 0Newell, David R.论文数: 0 引用数: 0 h-index: 0Noble, Martin E. M.论文数: 0 引用数: 0 h-index: 0Riedinger, Christiane论文数: 0 引用数: 0 h-index: 0Lunec, John论文数: 0 引用数: 0 h-index: 0Hardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0
- [8] Targeting the MDM2-p53 interaction: evaluation of a novel, potent MDM2-p53 antagonist in patient-derived CLL cellsLEUKEMIA & LYMPHOMA, 2020, 61 : 81 - 81论文数: 引用数: h-index:机构:Aptullahoglu, Erhan论文数: 0 引用数: 0 h-index: 0机构: Northern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, EnglandZhao, Yan论文数: 0 引用数: 0 h-index: 0机构: Northern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Newcastle Univ, Northern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, EnglandKyle, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England论文数: 引用数: h-index:机构:Ahn, Maria论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Pleasanton, CA USA Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, EnglandFazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Pleasanton, CA USA Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England论文数: 引用数: h-index:机构:Hardcastle, Ian论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, EnglandHoward, Steven论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Pleasanton, CA USA Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, EnglandChessari, Gianni论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Pleasanton, CA USA Newcastle Univ, Newcastle Upon Tyne, Tyne & Wear, England论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:
- [9] Energetic Landscape of MDM2-p53 Interactions by Computational Mutagenesis of the MDM2-p53 InteractionPLOS ONE, 2016, 11 (03):Thayer, Kelly M.论文数: 0 引用数: 0 h-index: 0机构: Dept Chem, 124 Raymond Ave, Poughkeepsie, NY 12604 USA Wesleyan Univ, Hall Atwater Labs, Middletown, CT 06459 USA Dept Chem, 124 Raymond Ave, Poughkeepsie, NY 12604 USABeyer, George A.论文数: 0 引用数: 0 h-index: 0机构: Vassar Coll, Biochem Program, 124 Raymond Ave, Poughkeepsie, NY 12604 USA Dept Chem, 124 Raymond Ave, Poughkeepsie, NY 12604 USA
- [10] Development of a potent class of small molecule inhibitors of the MDM2-p53 protein-protein interactionCANCER RESEARCH, 2018, 78 (13)Fazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandAhn, Maria论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandBevan, Luke论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandBuck, Ildiko论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandCastro, Juan论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandChessari, Gianni论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandCons, Ben论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandHearn, Keisha论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandHoward, Steven论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandJohnson, Chris论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandReeks, Judith论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandTamanini, Emiliano论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandThompson, Neil论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandWalton, Hugh论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandWilliams, Pamela论文数: 0 引用数: 0 h-index: 0机构: Astex Therapeut, Cambridge, England Astex Therapeut, Cambridge, EnglandBawn, Ruth H.论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandBlackburn, Tim J.论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandCano, Celine论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandCully, Sarah J.论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandGolding, Bernard论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandGriffin, Roger论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandHaggerty, Karen论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandHardcastle, Ian论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandNewell, Herbie论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandNoble, Martin论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandThomas, Huw论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandWillmore, Elaine论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandZhao, Yan论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, EnglandWedge, Steve论文数: 0 引用数: 0 h-index: 0机构: Nothern Inst Canc Res, Newcastle Upon Tyne, Tyne & Wear, England Astex Therapeut, Cambridge, England