共 29 条
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- [22] Synthesis and Biological Activity of 6-Substituted Pyrrolo[2,3-d]pyrimidine Thienoyl Regioisomers as Inhibitors of de Novo Purine Biosynthesis with Selectivity for Cellular Uptake by High Affinity Folate Receptors and the Proton-Coupled Folate Transporter over the Reduced Folate CarrierJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (04) : 1758 - 1770Wang, LeiCherian, ChristinaDesmoulin, Sita KugelMitchell-Ryan, ShermaineHou, ZhanjunMatherly, Larry H.Gangjee, Aleem
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- [27] Tumor-Targeting with Novel Non-Benzoyl 6-Substituted Straight Chain Pyrrolo[2,3-d]pyrimidine Antifolates via Cellular Uptake by Folate Receptor α and Inhibition of de Novo Purine Nucleotide BiosynthesisJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (21) : 8684 - 8695Wang, YiqiangCherian, ChristinaOrr, StevenMitchell-Ryan, ShermaineHou, ZhanjunRaghavan, SudhirMatherly, Larry H.Gangjee, Aleem
- [28] Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione Derivative Inhibits D-Dopachrome Tautomerase Activity and Suppresses the Proliferation of Non-Small Cell Lung Cancer CellsJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (03) : 2059 - 2077Xiao, ZhangpingOsipyan, AngelinaSong, ShanshanChen, DengSchut, Reinder A.van Merkerk, Ronaldvan der Wouden, Petra E.Cool, Robbert H.Quax, Wim J.Melgert, Barbro N.Poelarends, Gerrit J.Dekker, Frank J.
- [29] Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione Derivative Inhibits d-Dopachrome Tautomerase Activity and Suppresses the Proliferation of Non-Small Cell Lung Cancer Cells (vol 65, pg 2059, 2022)JOURNAL OF MEDICINAL CHEMISTRY, 2025, 68 (06) : 6844 - 6845Xiao, ZhangpingOsipyan, AngelinaSong, ShanshanChen, DengSchut, Reinder A.van Merkerk, Ronaldvan der Wouden, Petra E.Cool, Robbert H.Quax, Wim J.Melgert, Barbro N.Poelarends, Gerrit J.Dekker, Frank J.