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- [21] Structure-Based Design of an Iminoheterocyclic β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE) Inhibitor that Lowers Central Aβ in Nonhuman PrimatesJOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (07) : 3231 - 3248Mandal, Mihirbaran论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAWu, Yusheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAMisiaszek, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USALi, Guoqing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USABuevich, Alexei论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USACaldwell, John P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USALiu, Xiaoxiang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAMazzola, Robert D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAOrth, Peter论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAStrickland, Corey论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAVoigt, Johannes论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAWang, Hongwu论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAZhu, Zhaoning论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAChen, Xia论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAGrzelak, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAHyde, Lynn A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAKuvelkar, Reshma论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USALeach, Prescott T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USATerracina, Giuseppe论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAZhang, Lili论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAZhang, Qi论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAMichener, Maria S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Safety Assessment & Lab Anim Res, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USASmith, Brad论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Safety Assessment & Lab Anim Res, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USACox, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacokinet Pharmacodynam & Drug Metab, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAGrotz, Diane论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacokinet Pharmacodynam & Drug Metab, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAFavreau, Leonard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacokinet Pharmacodynam & Drug Metab, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAMitra, Kaushik论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacokinet Pharmacodynam & Drug Metab, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAKazakevich, Irina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Discovery Pharmaceut Sci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAMcKittrick, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAGreenlee, William论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAKennedy, Matthew E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAParker, Eric M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USACumming, Jared N.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USAStamford, Andrew W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Global Chem, 2015 Galloping Hill Rd, Kenilworth, NJ 07033 USA
- [22] Analysis of Natural Antisense Transcripts in Human beta-Site Amyloid Precursor Protein Cleaving Enzyme 1(BACE1)MODERN PATHOLOGY, 2009, 22 : 327A - 327AArai, C.论文数: 0 引用数: 0 h-index: 0机构: Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan Hirosaki Univ, Grad Sch Hlth Sci, Aomori, JapanMiura, T.论文数: 0 引用数: 0 h-index: 0机构: Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan Hirosaki Univ, Grad Sch Hlth Sci, Aomori, JapanKasai, K.论文数: 0 引用数: 0 h-index: 0机构: Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan Hirosaki Univ, Grad Sch Hlth Sci, Aomori, JapanNozaka, H.论文数: 0 引用数: 0 h-index: 0机构: Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan Hirosaki Univ, Grad Sch Hlth Sci, Aomori, JapanSato, T.论文数: 0 引用数: 0 h-index: 0机构: Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan Hirosaki Univ, Grad Sch Hlth Sci, Aomori, Japan
- [23] Structure-based design and synthesis of macroheterocyclic peptidomimetic inhibitors of the aspartic protease β-site amyloid precursor protein cleaving enzyme (BACE)JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (15) : 4544 - 4567Hanessian, Stephen论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, CanadaYang, Gaoqiang论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, CanadaRondeau, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, CanadaNeumann, Ulf论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, CanadaBetschart, Claudia论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, CanadaTintelnot-Blomley, Marina论文数: 0 引用数: 0 h-index: 0机构: Univ Montreal, Dept Chem, Montreal, PQ H3C 3J7, Canada
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- [25] Design and Synthesis of Potent, Orally Efficacious Hydroxyethylamine Derived β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE1) InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (21) : 9025 - 9044Dineen, Thomas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWeiss, Matthew M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWilliamson, Toni论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAActon, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USABabu-Khan, Safura论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USABrown, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAChen, Kui论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USACheng, Yuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USACitron, Martin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USACrogan, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USADunn, Robert T., II论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAEsmay, Joel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAGraceffa, Russell F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAHarriedt, Scott S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAHickman, Dean论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAHitchcock, Stephen A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAHorne, Daniel B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAHuang, Hongbing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAImbeah-Ampiah, Ronke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAJudd, Ted论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAKaller, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAKreiman, Charles R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USALa, Daniel S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USALi, Vivian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USALopez, Patricia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USALouie, Steven论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAMonenschein, Holger论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USANguyen, Thomas T.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAPennington, Lewis D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAMiguel, Tisha Sin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USASickmier, E. Allen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAVargas, Hugo M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWahl, Robert C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept HTS & Mol Pharmacol, Thousand Oaks, CA 91320 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWen, Paul H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWhittington, Douglas A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAWood, Stephen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAXue, Qiufen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAYang, Bryant H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAPatel, Vinod F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USAZhong, Wenge论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Chemica Res & Discovery, Cambridge, MA 02142 USA
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