SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF NEW 1,3-THIAZOLYLQUINAZOLIN-4-(3H)-ONES

被引：0

作者：

Patel, N. B. ^{[1
]}

Patel, J. N. ^{[1
]}

机构：

[1] Veer Narmad S Gujarat Univ, Dept Chem, Surat 395007, India

来源：

INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2009年 / 18卷 / 03期

关键词：

BIOLOGICAL EVALUATION; DERIVATIVES; ANTIBACTERIAL; AGENTS;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of 2-[2-(2,6-dichlorophenyl) amino] phenylmethyl-3-[4-substitutedanilino1,3-thiazol-2-yl]-6-iodoquinazolin-4-(3H) ones Va-o from 2-[(2,6-dichlorophenyl) amino]phenyl acetic acid I, via nucleophilic interaction of 2-[2-(2,6-dichlorophenyl) amino] phenylmethyl-6-iodo-3, 1-benzoxazin-4-(3H) ones III with thiourea nucleophile has been achieved. The final compounds have been characterized by analytical and spectral data (IR and H-1 NMR) and screened for their antimicrobial activity.

引用

页码：247 / 250

页数：4

共 18 条

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