Syntheses of Benzoimidazole Derivatives Containing Carbazole Unit

被引:5
|
作者
Bian, Lei [1 ]
Zeng, Xiangchao [1 ]
He, Ru [1 ]
Luo, Chuanglong [1 ]
Lin, Zhiqiang [1 ]
机构
[1] Jinan Univ, Dept Chem, Guangzhou 510632, Guangdong, Peoples R China
关键词
benzoimidazole; carbazole; organic synthesis; BENZIMIDAZOLE DERIVATIVES;
D O I
10.6023/cjoc201311018
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Two series of novel benzoimidazole derivatives containing carbazole unit were synthesized via condensation-cyclization of N-alkylcarbazole-3-formaldehyde with 1,2-diaminobenzene in "one pot" reaction without catalyst. The effects of temperature, selection & amount of solvents and molar ratio of the two reagents on the reactions have been investigated; significantly, one of these two series of benzoimidazole derivatives could be prepared as the major products selectively by changing the molar ratio of the two reagents.
引用
收藏
页码:994 / 998
页数:5
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