A convenient synthesis to N-aryl-substituted 4-piperidones

被引：15

作者：

Tortolani, DR ^{[1
]}

Poss, MA ^{[1
]}

机构：

[1] Bristol Myers Squibb Pharmaceut Res Inst, Combinatorial Drug Discovery, Princeton, NJ 08543 USA

来源：

ORGANIC LETTERS | 1999年 / 1卷 / 08期

关键词：

D O I：

10.1021/ol990930r

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[GRAPHICS] A general and efficient procedure for the synthesis of N-aryl-substituted 4-piperidones was developed. The general methodology was applied to the synthesis of several different N-aryl-4-piperidones utilizing an expedient two-step process.

引用

页码：1261 / 1262

页数：2

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