RELATIONSHIP OF PASSIVE PERMEABILITY AND CYTOCHROME P450 (CYP) 3A4 INHIBITION

被引：0
|
作者：
Li, Ling [1 ]
Zhou, Julia [1 ]
Nouraldeen, Amr [1 ]
Wilson, Alan G. E. [1 ]
机构：
[1] Lexicon Pharmaceut Inc, Dept DMPK Toxicol & Pathol, The Woodlands, TX USA
来源：
DRUG METABOLISM REVIEWS | 2014年 / 45卷
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：131 / 131
页数：1
相关论文
共 50 条
  • [1] Multivariate modeling of cytochrome P450 3A4 inhibition
    Kriegl, JM
    Eriksson, L
    Arnhold, T
    Beck, B
    Johansson, E
    Fox, T
    EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2005, 24 (05) : 451 - 463
  • [2] Inhibition of Human Cytochrome P450 3A4 by Cholesterol
    Shinkyo, Raku
    Guengerich, F. Peter
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2011, 286 (21) : 18426 - 18433
  • [3] Design and synthesis of a new fluorescent probe for cytochrome P450 3A4 (CYP 3A4)
    Chougnet, A
    Stoessel, C
    Woggon, WD
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (21) : 3643 - 3645
  • [4] Structures of cytochrome P450 3A4
    Scott, EE
    Halpert, JR
    TRENDS IN BIOCHEMICAL SCIENCES, 2005, 30 (01) : 5 - 7
  • [5] Development of cytochrome P450 3A4 inhibition model.
    Arimoto, R
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2004, 227 : U1019 - U1020
  • [6] QSAR modeling of in vitro inhibition of cytochrome P450 3A4*
    Mao, Boryeu
    Gozalbes, Rafael
    Barbosa, Frederique
    Migeon, Jacques
    Merrick, Sandra
    Kamm, Kelly
    Wong, Eric
    Costales, Chester
    Shi, Wei
    Wu, Cheryl
    Froloff, Nicolas
    JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2006, 46 (05) : 2125 - 2134
  • [7] Effect of cytochrome P450 3A4 inhibition on the pharmacokinetics of docetaxel
    Engels, FK
    ten Tije, AJ
    Baker, SD
    Lee, CKK
    Loos, WJ
    Vulto, AG
    Verweij, J
    Sparreboom, A
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 2004, 75 (05) : 448 - 454
  • [8] On the inhibition of cytochrome P450 3A4 by structurally diversified flavonoids
    Mitrasinovic, Petar M.
    JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2022, 40 (20): : 9713 - 9723
  • [9] Enantioselectivity of inhibition of cytochrome P450 3A4 (CYP3A4) by ketoconazole: Testosterone and methadone as substrates
    Dilmaghanian, S
    Gerber, JG
    Filler, SG
    Sanchez, A
    Gal, J
    CHIRALITY, 2004, 16 (02) : 79 - 85
  • [10] New fluorescent probes for Cytochrome P450 3A4 (CYP3A4)
    Chougnet, Antoinette
    JOURNAL OF BIOLOGICAL INORGANIC CHEMISTRY, 2007, 12 (SUPPL 1): : S55 - S55
12345