Novel diacid accelerated borane reducing agent for imines

被引：16

作者：

Lu, ZH ^{[1
]}

Bhongle, N ^{[1
]}

Su, XP ^{[1
]}

Ribe, S ^{[1
]}

Senanayake, CH ^{[1
]}

机构：

[1] Sepracor Inc, Chem Proc R&D, Marlborough, MA 01752 USA

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 47期

关键词：

reduction; imines; borane; diacids;

D O I：

10.1016/S0040-4039(02)01905-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A remarkable effect of diacids in modulating the reactivity of borane has been discovered. This novel process provides a rapid and excellent access for reduction of a variety of imines with different functionalities. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：8617 / 8620

页数：4

共 21 条

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