Discovery and characterization of covalent Pin1 inhibitors targeted to an active site cysteine

被引：0

作者：

Pinch, Benika ^{[1
]}

Doctor, Zainab ^{[2
,3
]}

Browne, Christopher M. ^{[2
,3
]}

Seo, Hyuk-Soo ^{[2
]}

Nabet, Behnam ^{[2
]}

Kozono, Shingo ^{[3
,4
]}

Lian, Xiaolan ^{[3
,4
]}

Zaidman, Daniel ^{[5
]}

Daitchman, Dina ^{[5
]}

London, Nir ^{[5
]}

Gong, Lu ^{[3
,4
]}

Manz, Theresa ^{[2
]}

Chun, Yujin ^{[3
]}

Tan, Li ^{[6
]}

Marto, Jarrod ^{[2
]}

Buratowski, Stephen ^{[3
]}

Dhe-Paganon, Sirano ^{[2
]}

Zhou, Xiao ^{[3
,4
]}

Lu, Kun Ping ^{[3
,4
]}

Gray, Nathanael S. ^{[2
,3
]}

机构：

[1] Harvard Univ, Cambridge, MA 02138 USA

[2] Dana Farber Canc Inst, Boston, MA 02115 USA

[3] Harvard Med Sch, Boston, MA 02115 USA

[4] Beth Israel Deaconess Med Ctr, Boston, MA 02215 USA

[5] Weizmann Inst Sci, Rehovot, Israel

[6] Chinese Acad Sci, Shanghai Inst Organ Chem, Shanghai, Peoples R China

来源：

CANCER RESEARCH | 2019年 / 79卷 / 13期

关键词：

D O I：

10.1158/1538-7445.AM2019-2757

中图分类号：

R73 [肿瘤学];

学科分类号：

100214 ;

摘要：

2757

引用

页数：2

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