Synthesis of ArSe-Substituted Flavone Derivatives Using Se Powder

被引：13

作者：

Feng, Chunlai ^{[1
]}

Zhu, Jie ^{[1
]}

Tang, Qiujie ^{[1
]}

Zhou, Aihua ^{[1
]}

机构：

[1] Jiangsu Univ, Pharm Sch, Zhenjiang 212013, Jiangsu, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2019年 / 39卷 / 04期

关键词：

selenium; C-Se bond; flavone; selenide; C-H functionalization; THIOETHERS; CHROMONES; SULFUR;

D O I：

10.6023/cjoc201808011

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

New flavone derivatives are highly valued in drug discovery due to their diversity of important bioactivities. Herein, one simple Cu-catalyzed method of constructing C-Se bonds on flavone structures using convenient Se powder via C-H functionalization is reported, regioselectively affording ArSe-substituted flavone derivatives in good yields.

引用

页码：1187 / 1192

页数：6

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