Design and synthesis of novel pyrrolo[2,1-c][1,4]benzodiazepine-imidazole containing polyamide conjugates

被引:0
作者
Kumar, R [1 ]
Reddy, BSN [1 ]
Lown, JW [1 ]
机构
[1] Univ Alberta, Dept Chem, Edmonton, AB T6G 2G2, Canada
关键词
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A series of novel pyrrolo[2,1-c][1,4]benzodiazepine(PBD)-polyamide conjugates (1-5) containing imidazole units was synthesized as DNA minor groove bining agents.
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页码:19 / 26
页数:8
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