Direct and catalytic synthesis of quinoxaline derivatives from epoxides and ene-1,2-diamines

被引:226
作者
Antoniotti, S
Duñach, E
机构
[1] Univ Nice, UMR CNRS 6001, Lab Aromes Synthese & Interact, Fac Sci, F-06108 Nice 2, France
[2] Univ Nice, UMR CNRS 6001, Chim Bioorgan Lab, Fac Sci, F-06108 Nice 2, France
关键词
quinoxaline; epoxides; heterocycles; bismuth; catalysis;
D O I
10.1016/S0040-4039(02)00715-3
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
We describe here a new synthesis of quinoxaline derivatives by a Bi-catalyzed oxidative coupling of epoxides and a ene-1.2-diamines. (C) 2002 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码:3971 / 3973
页数:3
相关论文
共 18 条
[1]   Bismuth(III) oxide perchlorate promoted rearrangement of epoxides to aldehydes and ketones [J].
Anderson, AM ;
Blazek, JM ;
Garg, P ;
Payne, BJ ;
Mohan, RS .
TETRAHEDRON LETTERS, 2000, 41 (10) :1527-1530
[2]   Novel and catalytic oxidation of internal epoxides to α-diketones [J].
Antoniotti, S ;
Duñach, E .
CHEMICAL COMMUNICATIONS, 2001, (24) :2566-2567
[3]  
BARLUENGA J, 1985, SYNTHESIS-STUTTGART, P313
[4]  
Brock E. D., 1999, [No title captured], Patent No. [WO 9951688, 9951688]
[5]  
Coin C, 2001, EUR J ORG CHEM, V2001, P735, DOI 10.1002/1099-0690(200102)2001:4<735::AID-EJOC735>3.0.CO
[6]  
2-E
[7]  
Dailey S, 2001, J MATER CHEM, V11, P2238, DOI 10.1039/b104674h
[8]  
EICHER T, 1995, CHEM HETEROCYCLES, P417
[9]   Tyrphostins .5. Potent inhibitors of platelet-derived growth factor receptor tyrosine kinase: Structure-activity relationships in quinoxalines, quinolines, and indole tyrphostins [J].
Gazit, A ;
App, H ;
McMahon, G ;
Chen, J ;
Levitzki, A ;
Bohmer, FD .
JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (11) :2170-2177
[10]  
Irwing-Sax N., 1989, DANGEROUS PROPERTIES, P283