First Conjugates of the Diterpenoid Isosteviol and Glucuronic Acid

被引：8

作者：

Andreeva, O. V. ^{[1
]}

Sharipova, R. R. ^{[1
]}

Strobykina, I. Yu. ^{[1
]}

Kataev, V. E. ^{[1
]}

机构：

[1] Russian Acad Sci, Kazan Sci Ctr, AE Arbuzov Organ & Phys Chem Inst, Kazan 420088, Russia

来源：

CHEMISTRY OF NATURAL COMPOUNDS | 2014年 / 50卷 / 03期

关键词：

isosteviol; diterpenes; diterpenoids; glucuronic acid; glucuronates; beyeranes; conjugates; CHEMICAL-SYNTHESIS; AMIDE DERIVATIVES; DELIVERY; AGENT; DRUG;

D O I：

10.1007/s10600-014-0988-7

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Conjugates of the diterpenoid isosteviol (16-oxo-ent-beyeran-19-oic acid) and glucuronic acid containing two diterpenoid (ent-beyerane) skeletons joined by a 1,6-hexanedicarboxylate spacer and beta-D-glucopyranuronoyl moieties were synthesized for the first time.

引用

页码：465 / 469

页数：5

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