A novel metal iodide promoted three-component synthesis of substituted pyrrolidines

被引：131
作者：
Bertozzi, F [1 ]
Gustafsson, M [1 ]
Olsson, R [1 ]
机构：
[1] ACADIA Pharmaceut AS, Discovery Chem, DK-2600 Glostrup, Denmark
来源：
ORGANIC LETTERS | 2002年 / 4卷 / 18期
关键词：
D O I：
10.1021/ol0264814
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[GRAPHICS] A new one-pot procedure for the synthesis of substituted pyrrolidine derivatives with commercially available cyclopropyl ketones, aldehydes, and amines by a metal iodide promoted three-component reaction was developed.
引用
收藏
页码：3147 / 3150
页数：4
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