One-pot Synthesis of Protected Alkylhydrazines from Acetals and Ketals. Scope and Limitations

被引：4

作者：

Mastitski, Anton ^{[1
]}

Niinepuu, Siret ^{[1
]}

Haljasorg, Toiv ^{[1
]}

Jaerv, Jaak ^{[1
]}

机构：

[1] Univ Tartu, Inst Chem, EE-50411 Tartu, Estonia

来源：

ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL | 2015年 / 47卷 / 06期

关键词：

SOLID-PHASE SYNTHESIS; PEPTIDE-SYNTHESIS; HYDRAZINE ALKYLATION; AMINO-ACIDS; AZA; DERIVATIVES; PRECURSORS; FMOC; AZAPEPTIDES; SCAN;

D O I：

10.1080/00304948.2015.1088760

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：490 / 498

页数：9

共 21 条

[1] Allais A., 1967, French Patent, Patent No. [1468633, 19671468633]
[2] Aza-amino acid scanning of secondary structure suited for solid-phase peptide synthesis with Fmoc chemistry and aza-amino acids with heteroatomic side chains
Boeglin, D
Lubell, WD
[J]. JOURNAL OF COMBINATORIAL CHEMISTRY, 2005, 7 (06): : 864 - 878
[3] Use of polyanions for alkylation of hydrazine derivatives
Bredihhin, Aleksei
Maeorg, Uno
[J]. ORGANIC LETTERS, 2007, 9 (24) : 4975 - 4977
[4] Solid-phase synthesis of "mixed" peptidomimetics using Fmoc-protected aza-/β3-amino acids and α-amino acids
Busnel, O
Bi, LR
Dali, H
Cheguillaume, A
Chevance, S
Bondon, A
Muller, S
Baudy-Floc'h, M
[J]. JOURNAL OF ORGANIC CHEMISTRY, 2005, 70 (26) : 10701 - 10708
[5] Preparation of new monomers aza-β3-aminoacids for solid-phase syntheses of aza-β3-peptides
Busnel, Olivier
Baudy-Floc'h, Michele
[J]. TETRAHEDRON LETTERS, 2007, 48 (33) : 5767 - 5770
[6] COISPEAU G, 1970, B SOC CHIM FR, P2717
[7] Aza-peptide analogs as potent human immunodeficiency virus type-1 protease inhibitors with oral bioavailability
Fassler, A
Bold, G
Capraro, HG
Cozens, R
Mestan, J
Poncioni, B
Rosel, J
TintelnotBlomley, M
Lang, M
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (16) : 3203 - 3216
[8] Microwave-Assisted Solid-Phase Aza-peptide Synthesis: Aza Scan of a PKB/Akt Inhibitor Using Aza-arginine and Aza-proline Precursors
Freeman, Noam S.
Tal-Gan, Yftah
Klein, Shoshana
Levitzki, Alexander
Gilon, Chaim
[J]. JOURNAL OF ORGANIC CHEMISTRY, 2011, 76 (09) : 3078 - 3085
[9] Synthesis of N′-substituted Ddz-protected hydrazines and their application in solid phase synthesis of aza-peptides
Freeman, Noam S.
Hurevich, Mattan
Gilon, Chaim
[J]. TETRAHEDRON, 2009, 65 (08) : 1737 - 1745
[10] Development of Near-Infrared Fluorophore (NIRF)-Labeled Activity-Based Probes for in Vivo Imaging of Legumain
Lee, Jiyoun
Bogyo, Matthew
[J]. ACS CHEMICAL BIOLOGY, 2010, 5 (02) : 233 - 243

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