Magnesiation of indoles with magnesium amide bases

被引：57

作者：

Kondo, Y

Yoshida, A

Sakamoto, T

机构：

[1] Faculty of Pharmaceutical Sciences, Tohoku University, Aobayama, Aoba-ku

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1996年 / 19期

关键词：

D O I：

10.1039/p19960002331

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-Substituted indole derivatives are deprotonated with Hauser bases (R(2)NMgBr) or magnesium diamide [(R(2)N)(2)Mg] to give magnesioindoles which are then reacted with electrophiles.

引用

页码：2331 / 2332

页数：2

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