A novel, chemically robust, amine releasing linker

被引：30

作者：

Kay, C

Murray, PJ

Sandow, L

Holmes, AB

机构：

[1] UNIV CAMBRIDGE,CHEM LABS,GLAXO WELLCOME CAMBRIDGE CHEM LAB,CAMBRIDGE CB2 1EW,ENGLAND

[2] UNIV CAMBRIDGE,CHEM LABS,DEPT CHEM,CAMBRIDGE CB2 1EW,ENGLAND

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 39期

关键词：

D O I：

10.1016/S0040-4039(97)01627-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A polymer supported sulfonamide 1, based on an amine protective group, has been developed as a novel linker for solid phase organic synthesis. The linker permits the immobilisation of alcohol substrates, and releases N-protected amines under mild nucleophilic cleavage conditions. (C) 1997 Elsevier Science Ltd.

引用

收藏

页码：6941 / 6944

页数：4

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