A medicinal chemistry perspective on artemisinin and related endoperoxides

[1] Predicting human oral bioavailability of a compound: Development of a novel quantitative structure-bioavailability relationship [J]. PHARMACEUTICAL RESEARCH, 2000, 17 (06) : 639 - 644

[2] [Anonymous], 2003, EUR J ORG CHEM, DOI DOI 10.1002/ejoc.200300064

[3] [Anonymous], INFECTION

[4] [Anonymous], 2002, DRUG METAB DISPOS

[5] REACTION OF ANTIMALARIAL ENDOPEROXIDES WITH SPECIFIC PARASITE PROTEINS [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1994, 38 (08) : 1854 - 1858

[6] Structure-activity relationships of the antimalarial agent artemisinin. 6. The development of predictive in vitro potency models using CoMFA and HQSAR methodologies [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (02) : 292 - 303

[7] Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (19) : 4321 - 4335

[8] SYNTHESIS, CONFORMATIONAL-ANALYSIS, AND ANTIMALARIAL ACTIVITY OF TRICYCLIC ANALOGS OF ARTEMISININ [J]. TETRAHEDRON, 1994, 50 (04) : 957 - 972

[9] Avery MA, 1996, J LABELLED COMPD RAD, V38, P263, DOI 10.1002/(SICI)1099-1344(199603)38:3&lt

[10] 263::AID-JLCR839&gt

[1] Predicting human oral bioavailability of a compound: Development of a novel quantitative structure-bioavailability relationship [J]. PHARMACEUTICAL RESEARCH, 2000, 17 (06) : 639 - 644

[2] [Anonymous], 2003, EUR J ORG CHEM, DOI DOI 10.1002/ejoc.200300064

[3] [Anonymous], INFECTION

[4] [Anonymous], 2002, DRUG METAB DISPOS

[5] REACTION OF ANTIMALARIAL ENDOPEROXIDES WITH SPECIFIC PARASITE PROTEINS [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1994, 38 (08) : 1854 - 1858

[6] Structure-activity relationships of the antimalarial agent artemisinin. 6. The development of predictive in vitro potency models using CoMFA and HQSAR methodologies [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (02) : 292 - 303

[7] Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2002, 45 (19) : 4321 - 4335

[8] SYNTHESIS, CONFORMATIONAL-ANALYSIS, AND ANTIMALARIAL ACTIVITY OF TRICYCLIC ANALOGS OF ARTEMISININ [J]. TETRAHEDRON, 1994, 50 (04) : 957 - 972

[9] Avery MA, 1996, J LABELLED COMPD RAD, V38, P263, DOI 10.1002/(SICI)1099-1344(199603)38:3&lt

[10] 263::AID-JLCR839&gt