SOLID-PHASE-BASED SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL CHROMOPHORE ANALOGUES OF THE BIS-INTERCALATOR TANDEM

被引:0
|
作者
Dawson, S. [1 ]
Searcey, M. [2 ]
Hampshire, A. [3 ]
Fox, K. [3 ]
Malkinson, J. [1 ]
机构
[1] Univ London, Sch Pharm, Dept Pharmaceut & Biol Chem, London WC1N 1AX, England
[2] Univ E Anglia, Sch Chem Sci & Pharm, Norwich NR4 7TJ, Norfolk, England
[3] Univ Southampton, Sch Biol Sci, Southampton SO16 7PX, Hants, England
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:367 / 367
页数:1
相关论文
共 50 条
  • [21] Synthesis and biological evaluation of novel epibatidine analogues.
    Cheng, J
    Zhang, CM
    Stevens, ED
    Izenwasser, S
    Wade, D
    Chen, SY
    Paul, D
    Trudell, ML
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 223 : A90 - A90
  • [22] Synthesis, biological evaluation and toxicity of novel tetrandrine analogues
    Schuetz, Ramona
    Mueller, Martin
    Geisslinger, Franz
    Vollmar, Angelika
    Bartel, Karin
    Bracher, Franz
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 207
  • [23] Synthesis and Biological Evaluation of Novel Gramicidin S Analogues
    Tuin, Adriaan Willem
    Palachanis, Dimitrios Konstantinos
    Buizert, Annelies
    Grotenbreg, Gijsbert Marnix
    Spalburg, Emile
    de Neeling, Albert J.
    Mars-Groenendijk, Roos H.
    Noort, Daan
    van der Marel, Gijsbert A.
    Overkleeft, Herman S.
    Overhand, Mark
    EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2009, 2009 (25) : 4231 - 4241
  • [24] Synthesis and biological evaluation of novel macrocyclic paclitaxel analogues
    Metaferia, BB
    Hoch, J
    Glass, TE
    Bane, SL
    Chatterjee, SK
    Snyder, JP
    Lakdawala, A
    Cornett, B
    Kingston, DGI
    ORGANIC LETTERS, 2001, 3 (16) : 2461 - 2464
  • [25] Synthesis and Biological Evaluation of Novel Bioisosteric Analogues of Dimebon™
    Ivachtchenko, Alexandre Vasilevich
    Frolov, Eugene Borisovich
    Mitkin, Oleg Dmitrievich
    Tkachenko, Sergey Evgenevich
    Khvat, Alexandre
    LETTERS IN DRUG DESIGN & DISCOVERY, 2010, 7 (06) : 446 - 451
  • [26] Solid-phase synthesis of acridine-based threading intercalator peptides
    Carlson, CB
    Beal, PA
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2000, 10 (17) : 1979 - 1982
  • [27] Solid-phase synthesis and biological evaluation of piperazine-based novel bacterial topoisomerase inhibitors
    Flagstad, Thomas
    Pedersen, Mette T.
    Jakobsen, Tim H.
    Felding, Jakob
    Tolker-Nielsen, Tim
    Givskov, Michael
    Qvortrup, Katrine
    Nielsen, Thomas E.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 57
  • [28] Synthesis and spectroscopic characterization of novel GFP chromophore analogues based on aminoimidazolone derivatives
    Jancso, Attila
    Kovacs, Ervin
    Cseri, Levente
    Rozsa, Balazs J.
    Galbacs, Gabor
    Csizmadia, Imre G.
    Mucsi, Zoltan
    SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY, 2019, 218 : 161 - 170
  • [29] Novel phthalimide based analogues: design, synthesis, biological evaluation, and molecular docking studies
    Othman, Ismail M. M.
    Gad-Elkareem, Mohamed A. M.
    El-Naggar, Mohamed
    Nossier, Eman S.
    Amr, Abd El-Galil E.
    JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2019, 34 (01) : 1259 - 1270
  • [30] Design, synthesis and evaluation of biological activity of novel fasudil analogues
    Li, Hang
    Wang, Donghua
    Liu, Shuai
    Sun, Changhai
    Chen, Meizhu
    Wang, Xinran
    Chen, Ligong
    PHARMAZIE, 2014, 69 (12): : 867 - 873