Traceless solid-phase organic synthesis

被引:146
作者
Blaney, P [1 ]
Grigg, R [1 ]
Sridharan, V [1 ]
机构
[1] Univ Leeds, Sch Chem, MIDAS Ctr, Leeds LS2 9JT, W Yorkshire, England
关键词
D O I
10.1021/cr0103827
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
An overview is given on the solid-phase synthesis of traceless organic compounds. Focus is on (a) traceless linkers, (b) miscellaneous traceless linkers, (c) cyclization-cleavage strategies in traceless synthesis, (d) traceless linkers for tertiary amine synthesis, and (e) traceless linkers for ureas, secondary amides, sulfonides, carbamates, and gaunidines.
引用
收藏
页码:2607 / 2624
页数:18
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