Structure-based design of Mcl-1 inhibitors: Interdiction at a protein-protein interface

被引:0
|
作者
Brown, Sean [1 ]
机构
[1] Amgen Inc, S San Fran, CA USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
202
引用
收藏
页数:1
相关论文
共 50 条
  • [41] Structure-based assessment and druggability classification of protein-protein interaction sites
    Alzyoud, Lara
    Bryce, Richard A.
    Al Sorkhy, Mohammad
    Atatreh, Noor
    Ghattas, Mohammad A.
    SCIENTIFIC REPORTS, 2022, 12 (01)
  • [42] A knowledge-based forcefield for protein-protein interface design
    Clark, Louis A.
    van Vlijmen, Herman W. T.
    PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2008, 70 (04) : 1540 - 1550
  • [43] Successful structure-based design of novel protein tyrosine phosphatase inhibitors
    Bower, Michael J.
    Combs, Andrew P.
    Yue, Eddy W.
    Ala, Paul J.
    Wayland, Brian
    Douty, Brent
    Takvorian, Amy
    Polam, Padmaja
    Wasserman, Zelda
    Zhu, Wenyu
    Crawley, Matthew
    Pruitt, James
    Sparks, Richard
    Glass, Brian
    Modi, Dilip
    McLaughlin, Erin
    Bostrom, Lori
    Li, Mei
    Galya, Laurine
    Blom, Karl
    Hillman, Milton
    Gonneville, Lucie
    Reid, Brian G.
    Wei, Min
    Becker-Pasha, Mary
    Klabe, Ronald
    Huber, Reid
    Li, Yanlong
    Hollis, Gregory
    Burn, Timothy C.
    Wynn, Richard
    Liu, Phillip
    Metcalf, Brian
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 231
  • [44] Structure-based design of protein-tyrosine phosphatase inhibitors.
    Burke, TR
    Yao, ZJ
    Ye, B
    Wang, SM
    Zhang, ZY
    Barford, D
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1997, 214 : 160 - COMP
  • [45] Protein-protein interface prediction based on hexagon structure similarity
    Guo, Fei
    Ding, Yijie
    Li, Shuai Cheng
    Shen, Chao
    Wang, Lusheng
    COMPUTATIONAL BIOLOGY AND CHEMISTRY, 2016, 63 : 83 - 88
  • [46] Structure-based design of protein-tyrosine phosphatase inhibitors.
    Moller, NPH
    Iversen, LF
    Hansen, TK
    Lau, J
    Petersen, AK
    Olsen, OH
    Moller, KB
    Mortensen, SB
    Billestrup, N
    Ge, Y
    Newman, MJ
    Holsworth, DD
    Lund, IK
    Andersen, B
    Peters, GH
    Andersen, HS
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 223 : B143 - B143
  • [47] Structure-based design and discovery of novel inhibitors of protein tyrosine phosphatases
    Huang, P
    Ramphal, J
    Wei, J
    Liang, CX
    Jallal, B
    McMahon, G
    Tang, C
    BIOORGANIC & MEDICINAL CHEMISTRY, 2003, 11 (08) : 1835 - 1849
  • [48] STRUCTURE-BASED DESIGN OF SELECTIVE INHIBITORS AGAINST THE BACE PROTEIN FAMILY
    Lendy, Emma
    Cardenas, Emilio
    Yen, Yu-Chen
    Ghosh, Arun
    Mesecar, Andrew
    PROTEIN SCIENCE, 2019, 28 : 189 - 189
  • [49] In silico design of potential Mcl-1 peptide-based inhibitors
    Faraji, Naser
    Daly, Norelle L.
    Arab, Seyed Shahriar
    Khosroushahi, Ahmad Yari
    JOURNAL OF MOLECULAR MODELING, 2024, 30 (04)
  • [50] In silico design of potential Mcl-1 peptide-based inhibitors
    Naser Faraji
    Norelle L. Daly
    Seyed Shahriar Arab
    Ahmad Yari Khosroushahi
    Journal of Molecular Modeling, 2024, 30