共 50 条
- [31] Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein-Protein InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (07) : 4071 - 4088Chessari, Gianni论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAhn, Jong Sook论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAnil, Burcu论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAnscombe, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBawn, Ruth H.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBevan, Luke D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBlackburn, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBuck, Ildiko论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCano, Celine论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCarbain, Benoit论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCastro, Juan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCons, Ben论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCully, Sarah J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandEndicott, Jane A.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandFazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandGolding, Bernard T.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandGriffin, Roger J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHaggerty, Karen论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHarnor, Suzannah J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHearn, Keisha论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHobson, Stephen论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHolvey, Rhian S.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHoward, Steven论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandJennings, Claire E.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandJohnson, Christopher N.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, England论文数: 引用数: h-index:机构:Miller, Duncan C.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandNewell, David R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandNoble, Martin E. M.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandReeks, Judith论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandRevill, Charlotte H.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandRiedinger, Christiane论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandSt Denis, Jeffrey D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandTamanini, Emiliano论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandThomas, Huw论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandThompson, Neil T.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandVinkovic, Mladen论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWedge, Stephen R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWilliams, Pamela A.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWilsher, Nicola E.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandZhang, Bian论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandZhao, Yan论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, England
- [32] Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 InhibitorsACS MEDICINAL CHEMISTRY LETTERS, 2017, 8 (02): : 239 - 244Johannes, Jeffrey W.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USABates, Stephanie论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Cambridge, Sci Pk,Unit 310 Darwin Bldg, Cambridge CB4 0WGD, England AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USABeigie, Carl论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA Sanofi Genzyme, Off 3216A C 3, One Res Dr, Westborough, MA 01581 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USABelmonte, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USABreen, John论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA Fdn Med Inc, 150 Second St, Cambridge, MA 02141 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USACao, Shenggen论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USACentrella, Paolo A.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAClark, Matthew A.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USACuozzo, John W.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USADumelin, Christoph E.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA Novartis Pharma AG, Novartis Inst Biomed Res, Basel, Switzerland AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAFerguson, Andrew D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAHabeshian, Sevan论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA Fulcrum Therapeut, One Kendall Sq,Bldg 700,Suite B7102, Cambridge, MA 02139 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAHargreaves, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAJoubran, Camil论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA Alkermes Inc, 852 Winter St, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAKazmirski, Steven论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAKeefe, Anthony D.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USALamb, Michelle L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USALan, Haiye论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USALi, Yunxia论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAMa, Hao论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAMlynarski, Scott论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAPacker, Martin J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Alderley Pk, Macclesfield SK10 4TG, Cheshire, England AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USARawlins, Philip B.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Cambridge, Sci Pk,Unit 310 Darwin Bldg, Cambridge CB4 0WGD, England AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USARobbins, Daniel W.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA Nurix Inc, 1700 Owens St,Suite 290, San Francisco, CA 94158 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAShen, Haidong论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USASigel, Eric A.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USASoutter, Holly H.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USASu, Nancy论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USATroast, Dawn M.论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA Morph Therapeut Inc, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAWang, Haiyun论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAWickson, Kate F.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAWu, Chengyan论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAZhang, Ying论文数: 0 引用数: 0 h-index: 0机构: X Chem Pharmaceut, 100 Beaver St, Waltham, MA 02453 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAZhao, Qiuying论文数: 0 引用数: 0 h-index: 0机构: Pharmaron Beijing Co Ltd, 6 Taihe Rd BDA, Beijing 100176, Peoples R China AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAZheng, Xiaolan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USAHird, Alexander W.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA AstraZeneca R&D Boston, 35 Gatehouse Dr, Waltham, MA 02451 USA
- [33] Structure-Based Design of Non-natural Macrocyclic Peptides That Inhibit Protein-Protein InteractionsJOURNAL OF MEDICINAL CHEMISTRY, 2017, 60 (21) : 8982 - 8988Krueger, Dennis M.论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany TU Dortmund Univ, Fac Chem & Chem Biol, Otto Hahn Str 6, D-44227 Dortmund, Germany Uppsala Univ, Dept Cell & Mol Biol, BMC Box 596, S-75124 Uppsala, Sweden Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyGlas, Adrian论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany TU Dortmund Univ, Fac Chem & Chem Biol, Otto Hahn Str 6, D-44227 Dortmund, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyBier, David论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany Univ Duisburg Essen, Dept Chem, Univ Str 7, D-45141 Essen, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyPospiech, Nicole论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyWallraven, Kerstin论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyDietrich, Laura论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany TU Dortmund Univ, Fac Chem & Chem Biol, Otto Hahn Str 6, D-44227 Dortmund, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany论文数: 引用数: h-index:机构:Koch, Oliver论文数: 0 引用数: 0 h-index: 0机构: TU Dortmund Univ, Fac Chem & Chem Biol, Otto Hahn Str 6, D-44227 Dortmund, Germany Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyHennig, Sven论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany Vrije Univ Amsterdam, Dept Chem & Pharmaceut Sci, De Boelelaan 1083, NL-1081 HV Amsterdam, Netherlands Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, GermanyGrossmann, Tom N.论文数: 0 引用数: 0 h-index: 0机构: Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany TU Dortmund Univ, Fac Chem & Chem Biol, Otto Hahn Str 6, D-44227 Dortmund, Germany Vrije Univ Amsterdam, Dept Chem & Pharmaceut Sci, De Boelelaan 1083, NL-1081 HV Amsterdam, Netherlands Max Planck Gesell, Chem Genom Ctr, Otto Hahn Str 15, D-44227 Dortmund, Germany
- [34] Structure-based design of a protein-protein interaction inhibitor, ABT-263, for the treatment of cancerABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Wendt, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA
- [35] Structure-based design of N-substituted 1-hydroxy-4-sulfamoyl-2naphthoates as selective inhibitors of the Mcl-1 oncoproteinEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 113 : 273 - 292Lanning, Maryanna E.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAYu, Wenbo论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAYap, Jeremy L.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAChauhan, Jay论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAChen, Lijia论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAWhiting, Ellis论文数: 0 引用数: 0 h-index: 0机构: Cardiff Univ, Sch Chem, Cardiff CF10 3AT, S Glam, Wales Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAPidugu, Lakshmi S.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Med, Ctr Biomol Therapeut, Dept Biochem & Mol Biol, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAAtkinson, Tyler论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, PharmD Program, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USABailey, Hala论文数: 0 引用数: 0 h-index: 0机构: Bryn Mawr Sch, 109 W Melrose Ave, Baltimore, MD 21210 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USALi, Willy论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, PharmD Program, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USARoth, Braden M.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Med, Ctr Biomol Therapeut, Dept Biochem & Mol Biol, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAHynicka, Lauren论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharm Practice & Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAChesko, Kirsty论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAToth, Eric A.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Med, Ctr Biomol Therapeut, Dept Biochem & Mol Biol, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAShapiro, Paul论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAMacKerell, Alexander D., Jr.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAWilder, Paul T.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Med, Ctr Biomol Therapeut, Dept Biochem & Mol Biol, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USAFletcher, Steven论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA Univ Maryland, Greenebaum Canc Ctr, 22 S Greene St, Baltimore, MD 21201 USA Univ Maryland, Sch Pharm, Dept Pharmaceut Sci, 20 N Pine St, Baltimore, MD 21201 USA
- [36] Design of Protein-Protein Interaction Inhibitors Based on Protein Epitope MimeticsCHEMBIOCHEM, 2009, 10 (06) : 971 - 973Robinson, John A.论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Dept Chem, CH-8057 Zurich, Switzerland Univ Zurich, Dept Chem, CH-8057 Zurich, Switzerland
- [37] Fragment-based discovery of potent inhibitors of the anti-apoptotic MCL-1 proteinBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (06) : 1484 - 1488Petros, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USASwann, Steven L.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USASong, Danying论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USASwinger, Kerren论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USAPark, Chang论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USAZhang, Haichao论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USAWendt, Michael D.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USAKunzer, Aaron R.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USASouers, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USASun, Chaohong论文数: 0 引用数: 0 h-index: 0机构: AbbVie, Res & Dev, N Chicago, IL 60064 USA AbbVie, Res & Dev, N Chicago, IL 60064 USA
- [38] Protein-Protein Interaction Prediction via Structure-Based Deep LearningPROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2024, 92 (11) : 1287 - 1296Liu, Yucong论文数: 0 引用数: 0 h-index: 0机构: Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R China Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R ChinaLiu, Yijun论文数: 0 引用数: 0 h-index: 0机构: Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R China Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R ChinaLi, Zhenhai论文数: 0 引用数: 0 h-index: 0机构: Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R China Shanghai Univ, Shanghai Inst Appl Math & Mech, Sch Mech & Engn Sci, Shanghai Key Lab Mech Energy Engn, Shanghai, Peoples R China
- [39] Structure-based de novo design of selective inhibitors for beta-catenin/Tcf protein-protein interactions in the Wnt signaling pathwayABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243Huang, Zheng论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Dept Chem, Salt Lake City, UT 84112 USA Univ Utah, Ctr Cell & Genome Sci, Salt Lake City, UT 84112 USA Univ Utah, Dept Chem, Salt Lake City, UT 84112 USAYu, Binxun论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Dept Chem, Salt Lake City, UT 84112 USA Univ Utah, Ctr Cell & Genome Sci, Salt Lake City, UT 84112 USA Univ Utah, Dept Chem, Salt Lake City, UT 84112 USAZhang, Min论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Dept Chem, Salt Lake City, UT 84112 USA Univ Utah, Ctr Cell & Genome Sci, Salt Lake City, UT 84112 USA Univ Utah, Dept Chem, Salt Lake City, UT 84112 USAJi, Haitao论文数: 0 引用数: 0 h-index: 0机构: Univ Utah, Dept Chem, Salt Lake City, UT 84112 USA Univ Utah, Ctr Cell & Genome Sci, Salt Lake City, UT 84112 USA Univ Utah, Dept Chem, Salt Lake City, UT 84112 USA
- [40] Comparison of Sequence-and Structure-Based Protein-Protein Interaction Sites2016 IEEE EMBS INTERNATIONAL STUDENT CONFERENCE (ISC), 2016,Dick, Kevin论文数: 0 引用数: 0 h-index: 0机构: Carleton Univ, Syst & Comp Engn, Ottawa, ON, Canada Carleton Univ, Syst & Comp Engn, Ottawa, ON, Canada论文数: 引用数: h-index:机构: