共 50 条
- [1] Selective and Potent Morpholinone Inhibitors of the MDM2-p53 Protein-Protein InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2014, 57 (06) : 2472 - 2488Gonzalez, Ana Z.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAEksterowicz, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USABeck, Hilary P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAChow, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USADuquette, Jason论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAFox, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAFu, Jiasheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAHouze, Jonathan B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAJin, Lixia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALi, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALi, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALing, Yun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USALong, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcGee, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcIntosh, Joel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMcMinn, Dustin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USARew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAShaffer, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAWortman, Sarah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYakowec, Peter论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAOlson, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, 1120 Vet Blvd, San Francisco, CA 94080 USA
- [2] Identification of substituted isoindolinones as potent inhibitors of the MDM2-p53 protein-protein interactionMOLECULAR CANCER THERAPEUTICS, 2009, 8 (12)Watson, Anna论文数: 0 引用数: 0 h-index: 0Liu, Junfeng论文数: 0 引用数: 0 h-index: 0Armstrong, Elizabeth论文数: 0 引用数: 0 h-index: 0Blackburn, Timothy论文数: 0 引用数: 0 h-index: 0Endicott, Jane A.论文数: 0 引用数: 0 h-index: 0Golding, Bernard T.论文数: 0 引用数: 0 h-index: 0Griffin, Roger J.论文数: 0 引用数: 0 h-index: 0Lu, Xiaohong论文数: 0 引用数: 0 h-index: 0Newell, David R.论文数: 0 引用数: 0 h-index: 0Noble, Martin E. M.论文数: 0 引用数: 0 h-index: 0Riedinger, Christiane论文数: 0 引用数: 0 h-index: 0Lunec, John论文数: 0 引用数: 0 h-index: 0Hardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0
- [3] Small-molecule inhibitors of the MDM2-p53 protein-protein interaction based on an isoindolinone scaffoldJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (21) : 6209 - 6221Hardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAhmed, Shafiq U.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAtkins, Helen论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandFarnie, Gillian论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGolding, Bernard T.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGriffin, Roger J.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGuyenne, Sabrina论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandHutton, Claire论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKallblad, Per论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKemp, Stuart J.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKitching, Martin S.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNewell, David R.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNorbedo, Stefano论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNorthen, Julian S.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandReid, Rebecca J.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandSaravanan, K.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandWillems, Henriette M. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandLunec, John论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, No Inst Canc Res, Sch Nat Sci Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England
- [4] Discovery of MDM2-p53 and MDM4-p53 protein-protein interactions small molecule dual inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 241Espadinha, Margarida论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalLopes, Elizabeth A.论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalMarques, Vanda论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalAmaral, Joana D.论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugaldos Santos, Daniel J. V. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Lusofona Humanidades & Tecnol, Res Ctr Biosci & Hlth Technol, CBIOS, P-1749024 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalMori, Mattia论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dept Biotechnol Chem & Pharm, Via Aldo Moro 2, I-53100 Siena, Italy Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal论文数: 引用数: h-index:机构:Piccarducci, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalZappelli, Elisa论文数: 0 引用数: 0 h-index: 0机构: Univ Pisa, Dept Pharm, I-56126 Pisa, Italy Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal论文数: 引用数: h-index:机构:Rodrigues, Cecilia M. P.论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, PortugalSantos, Maria M. M.论文数: 0 引用数: 0 h-index: 0机构: Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, iMed ULisboa Fac Pharm, Med Organ Chem Grp, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal Univ Lisbon, Res Inst Med iMed ULisboa, Fac Pharm, Ave Prof Gama Pinto, P-1649003 Lisbon, Portugal
- [5] Discovery of sulfonamide-piperidinones as potent inhibitors of the MDM2-p53 protein-protein interactionCANCER RESEARCH, 2015, 75Li, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAFu, Jiasheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USARew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAGribble, Michael W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, San Francisco, CA USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAEksterowicz, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA USA Amgen Inc, San Francisco, CA USAJin, Lixia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAMcGee, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, San Francisco, CA USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, San Francisco, CA USAShaffer, Paul论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Cambridge, MA USA Amgen Inc, San Francisco, CA USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAWortman, Sarah论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, San Francisco, CA USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, San Francisco, CA USAOlson, Steve H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USA
- [6] Small-Molecule Inhibitors of the MDM2-p53 Protein-Protein Interaction (MDM2 Inhibitors) in Clinical Trials for Cancer TreatmentJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (03) : 1038 - 1052Zhao, Yujun论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAAguilar, Angelo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USABernard, Denzil论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
- [7] Isoindolinone based inhibitors of the MDM2-p53 protein-protein interactionABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2735 - U2736Kemp, SJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandHardcastle, IR论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAhmed, SU论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAtatreh, NA论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandBarrett, P论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandEndicott, JA论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGolding, BT论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGriffin, RJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGruber, J论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandHutton, C论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England论文数: 引用数: h-index:机构:Noble, MEM论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandReid, RJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandRiedinger, C论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandSmyth, LA论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Univ Newcastle Upon Tyne, Sch Nat Sci, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England
- [8] Small molecule protein-protein inhibitors for the p53-MDM2 interactionCURRENT TOPICS IN MEDICINAL CHEMISTRY, 2007, 7 (10) : 952 - 960Dudkina, Anna S.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALindsley, Craig W.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA
- [9] The development of piperidinones as potent MDM2-P53 protein - protein interaction inhibitors for cancer therapyEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 159 : 1 - 9Liao, Guochao论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaYang, Deying论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaMa, Leilei论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaLi, Wenwei论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaHu, Liqin论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaZeng, Liming论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaWu, Peng论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaDuan, Lixin论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R ChinaLiu, Zhongqiu论文数: 0 引用数: 0 h-index: 0机构: Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China Guangzhou Univ Chinese Med, Joint Lab Translat Canc Res Chinese Med, Minist Educ Peoples Republ China, Int Inst Translat Chinese Med, Guangzhou 510006, Guangdong, Peoples R China
- [10] Isoindolinone-based inhibitors of the MDM2-p53 protein-protein interactionBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (05) : 1515 - 1520Hardcastle, IR论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAhmed, SU论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandAtkins, H论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandCalvert, AH论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandCurtin, NJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandFarnie, G论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGolding, BT论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGriffin, RJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandGuyenne, S论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandHutton, C论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKällbad, P论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKemp, SJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandKitching, MS论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNewell, DR论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNorbedo, S论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandNorthen, JS论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandReid, RJ论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandSaravanan, K论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandWillems, HMG论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, EnglandLunec, J论文数: 0 引用数: 0 h-index: 0机构: Univ Newcastle Upon Tyne, Sch Nat Sci Chem, No Inst Canc Res, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England