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- [31] The Discovery of Polo-Like Kinase 4 Inhibitors: Identification of (1R,2S)-2-(3((E)-4-(((cis)-2,6-Dimethylmorpholino)methyl)styryl)-1H-indazol-6-yl)-5′-methoxyspiro[cyclopropane-1,3′-indolin]-2′-one (CFI-400945) as a Potent, Orally Active Antitumor AgentJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (01) : 147 - 169Sampson, Peter B.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaLiu, Yong论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaForrest, Bryan论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaCumming, Graham论文数: 0 引用数: 0 h-index: 0机构: Celt Catalysts, Nova Ctr 1 03, Dublin 4, Ireland Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaLi, Sze-Wan论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaPatel, Narendra Kumar论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaEdwards, Louise论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaLaufer, Radoslaw论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaFeher, Miklos论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaBan, Fuqiang论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaAwrey, Donald E.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaMao, Guodong论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaPlotnikova, Olga论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaHodgson, Richard论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaBeletskaya, Irina论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaMason, Jacqueline M.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaLuo, Xunyi论文数: 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Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaHuang, Ping论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaMak, Tak W.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaPan, Guohua论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, CanadaPauls, Henry W.论文数: 0 引用数: 0 h-index: 0机构: Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada Univ Hlth Network, MaRS Ctr, Campbell Family Inst Breast Canc Res, Toronto, ON MG5 1L7, Canada
- [32] Discovery of (2S)-8[(3R)-3-Methylmorpholin-4-yl]-1-(3-methyl-2-oxobutyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido[1,2-a]pyrimidin-6-one: A Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid TumorsJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (01) : 376 - 400Pasquier, Benoit论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceEl-Ahmad, Youssef论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceFiloche-Romme, Bruno论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceDureuil, Christine论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceFassy, Florence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceAbecassis, Pierre-Yves论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Drug Disposit & Safety, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMathieu, Magali论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBertrand, Thomas论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBenard, Tsiala论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Pharmaceut Sci Operat, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBarriere, Cedric论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceEl Batti, Samira论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLetallec, Jean-Philippe论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceSonnefraud, Veronique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBrollo, Maurice论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceDelbarre, Laurence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLoyau, Veronique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FrancePilorge, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBertin, Luc论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceRichepin, Patrick论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceArigon, Jerome论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceLabrosse, Jean-Robert论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 Montpellier, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceClement, Jacques论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Lead Generat Candidate Realizat LGCR C&BD, F-34184 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h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceBretin, Francois论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMarquette, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Struct Design Informat & Struct Biol, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceMichot, Nadine论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Prot Prod, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceCaron, Anne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Global Biotherapeut, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceCastell, Christelle论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, France Sanofi, Oncol Drug Discovery, F-94403 Vitry Sur Seine, FranceSchio, Laurent论文数: 0 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- [33] Discovery of 2-(2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino [2′,3′:3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitorBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (24) : 5977 - 5984Muthukaman, Nagarajan论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaDeshmukh, Sanjay论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaSarode, Neelam论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaTondlekar, Shital论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaTambe, Macchindra论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaPisal, Dnyandeo论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaShaikh, Mahamadhanif论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaKattige, Vidya G.论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaHonnegowda, Srinivasa论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaKarande, Vikas论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaKulkarni, Abhay论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaJadhav, Satyawan B.论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaMahat, Mahamad Yunnus A.论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaGudi, Girish S.论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Drug Metab & Pharmacokinet, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaKhairatkar-Joshi, Neelima论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Biol Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, IndiaGharat, Laxmikant A.论文数: 0 引用数: 0 h-index: 0机构: Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India Glenmark Pharmaceut Ltd, Glenmark Res Ctr, Chem Res, Navi Mumbai 400709, Maharashtra, India
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