Multicomponent synthesis of nicotinic acid derivatives

被引：5

作者：

Dyachenko, Ivan V. ^{[1
]}

Dyachenko, Vladimir D. ^{[1
]}

Dorovatovskii, Pavel V. ^{[2
]}

Khrustalev, Victor N. ^{[3
,4
]}

Nenajdenko, Valentine G. ^{[5
]}

机构：

[1] Luhansk Taras Shevchenko Natl Univ, 2 Oboronna St, UA-91000 Lugansk, Ukraine

[2] Kurchatov Inst, Natl Res Ctr, 1 Akad Kurchatova Sq, Moscow 123182, Russia

[3] RUDN Univ, 6 Miklukho Maklaya St, Moscow 117198, Russia

[4] Russian Acad Sci, ND Zelinsky Inst Organ Chem, 47 Leninsky Ave, Moscow 119991, Russia

[5] Lomonosov Moscow State Univ, 1,Build 3 Leninskie Gory, Moscow 119991, Russia

来源：

CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2020年 / 56卷 / 12期

关键词：

6-alkoxy-2-alkylsulfanyl-4-methyl(4,4-dimethyl)nicotinic acid; CH acids; thiazolo[3,2-a]pyridines; alkylation; Michael reaction; multicomponent synthesis; X-ray structural analysis;

D O I：

10.1007/s10593-020-02852-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of previously unknown nitriles, esters, and an amide of 6-alkoxy-2-alkylsulfanyl-4-methyl(4,4-dimethyl)nicotinic acid has been developed. The structure of a number of the obtained derivatives was proved by X-ray structural analysis.

引用

页码：1579 / 1585

页数：7

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