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- [22] Novel Allosteric Mechanism of Dual p53/MDM2 and p53/MDM4 Inhibition by a Small MoleculeFRONTIERS IN MOLECULAR BIOSCIENCES, 2022, 9Grinkevich, Vera V.论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenVema, Aparna论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Chem, Div Organ Pharmaceut Chem, Uppsala, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenFawkner, Karin论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenIssaeva, Natalia论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Dept Otolaryngol Head & Neck Surg, Chapel Hill, NC USA Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenAndreotti, Virginia论文数: 0 引用数: 0 h-index: 0机构: IRCCS Osped Policlin San Martino, Genet Rare Canc, Genoa, Italy Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenDickinson, Eleanor R.论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Manchester Inst Biotechnol, Sch Chem, Manchester, England Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenHedstrom, Elisabeth论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenSpinnler, Clemens论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenInga, Alberto论文数: 0 引用数: 0 h-index: 0机构: Univ Trento, Dept CIBIO, Trento, Italy Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenLarsson, Lars-Gunnar论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenKarlen, Anders论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Med Chem, Div Organ Pharmaceut Chem, Uppsala, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenWilhelm, Margareta论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenBarran, Perdita E.论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Manchester Inst Biotechnol, Sch Chem, Manchester, England Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenOkorokov, Andrei L.论文数: 0 引用数: 0 h-index: 0机构: UCL, Wolfson Inst Biomed Res, London, England Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenSelivanova, Galina论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, SwedenZawacka-Pankau, Joanna E.论文数: 0 引用数: 0 h-index: 0机构: Karolinska Inst, Ctr Hematol & Regenerat Med, Dept Med, Huddinge, Stockholm, Sweden Karolinska Inst, Dept Microbiol, Tumor & Cell Biol, Stockholm, Sweden
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- [24] KT-253, a Novel MDM2 Degrader and p53 Stabilizer, Has Superior Potency and Efficacy than MDM2 Small-Molecule InhibitorsMOLECULAR CANCER THERAPEUTICS, 2025, 24 (04) : 497 - 510Chutake, Yogesh K.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAMayo, Michele F.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USADumont, Nancy论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAFiliatrault, Jessica论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USABreitkopf, Susanne B.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USACho, Patricia论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAChen, Dapeng论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USADixit, Vaishali S.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAProctor, William R.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAKuhn, Eric W.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAMartinez, Sarah Bollinger论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAMcdonald, Alice A.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAQi, Jianfeng论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAHu, Kan-Nian论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAKarnik, Rahul论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAGrowney, Joseph D.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USASharma, Kirti论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USASchalm, Stefanie S.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAGollerkeri, Ashwin M.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAMainolfi, Nello论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAWilliams, Juliet A.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USAWeiss, Matthew M.论文数: 0 引用数: 0 h-index: 0机构: Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA Kymera Therapeut Inc, 500 North Beacon St, Watertown, MA 02472 USA
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